SCHEMBL7607637

SCHEMBL7607637

COC(=O)Nc1ccc(C(CCNC[C@H](O)COc2ccc(OCc3ccccc3)c(N)c2)c2ccc(N(Cc3ccccc3)C(=O)OC)cc2)cc1

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 11/20 0.42
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
MEN1 O00255 1/20 0.40
OPRM1 P35372 1/20 0.40
OPRD1 P41143 1/20 0.40
KMT2A Q03164 1/20 0.40
ADRB1 P08588 7/20 0.40
ADRB3 P13945 7/20 0.40
ADRB2 P07550 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7536025 0.91 NPC1 (0.51) ABCB1NPC1RAB9ASMN1; SMN2MEN1
SCHEMBL7612154 0.89 NPC1 (0.39) NPC1RAB9ASMN1; SMN2MEN1KMT2A
SCHEMBL7609851 0.89 NPC1 (0.39) NPC1RAB9ASMN1; SMN2MEN1KMT2A
SCHEMBL7597017 0.88 MEN1 (0.53) ABCB1MEN1OPRM1OPRD1KMT2A
SCHEMBL7605875 0.81 ADRB1 (0.46) NPC1RAB9ASMN1; SMN2ADRB1ADRB3
SCHEMBL7610964 0.81 NPC1 (0.46) ABCB1NPC1RAB9ASMN1; SMN2
SCHEMBL6322792 0.81 NPC1 (0.46) ABCB1NPC1RAB9ASMN1; SMN2
SCHEMBL7612353 0.80 NPC1 (0.48) ABCB1NPC1RAB9ASMN1; SMN2
SCHEMBL6327240 0.76 MEN1 (0.70) ABCB1MEN1OPRM1OPRD1KMT2A
SCHEMBL7033981 0.76 MEN1 (0.70) ABCB1MEN1OPRM1OPRD1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1230210-A1 AMINOALCOHOL DERIVATIVES USEFUL FOR THE TREATMENT OF GASTROINTESTINAL DISORDERS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2002-08-14 EP disclosed
EP-1107944-A1 AMINOALCOHOL DERIVATIVES AND THEIR USE AS BETA 3 ADRENERGIC AGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-06-20 EP disclosed
WO-2001036375-A1 AMINOALCOHOL DERIVATIVES USEFUL FOR THE TREATMENT OF GASTROINTESTINAL DISORDERS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-05-25 WO disclosed
WO-2000012462-A1 AMINOALCOHOL DERIVATIVES AND THEIR USE AS BETA 3 ADRENERGIC AGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-03-09 WO disclosed