SCHEMBL7610643

SCHEMBL7610643

O=C(NCNC(=O)c1ccccc1C(=O)c1ccccc1)Nc1cccc(C(=O)OCc2ccccc2)c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 3/20 0.58
KMT2A Q03164 4/20 0.47
MEN1 O00255 3/20 0.47
ALDH1A1 P00352 3/20 0.46
CYP2C9 P11712 2/20 0.46
CYP2C19 P33261 2/20 0.46
NPSR1 Q6W5P4 2/20 0.46
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
POLB P06746 2/20 0.46
PKM P14618 1/20 0.46
MAPT P10636 5/20 0.46
PPIA P62937 2/20 0.46
THRB P10828 1/20 0.46
SLC6A2 P23975 1/20 0.45
SLC6A3 Q01959 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
HTT P42858 2/20 0.44
NAMPT P43490 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7610763 0.86 RAB9A (0.47) RAB9AKMT2AMEN1ALDH1A1CYP3A4
SCHEMBL20442339 0.81 RAB9A (0.78) RAB9AKMT2AMEN1ALDH1A1POLB
SCHEMBL8669488 0.80 RAB9A (0.69) RAB9AKMT2AMEN1ALDH1A1CYP2C9
SCHEMBL8130235 0.79 RAB9A (0.67) RAB9AKMT2AMEN1ALDH1A1CYP2C9
SCHEMBL27471805 0.75 RAB9A (0.76) RAB9AKMT2AALDH1A1CYP2C9CYP2C19
SCHEMBL8683973 0.74 RAB9A (0.75) RAB9AKMT2AMEN1ALDH1A1CYP2C9
Hydrochloric Acid SCHEMBL27455337 0.74 RAB9A (0.74) RAB9AKMT2AALDH1A1CYP2C9CYP2C19
SCHEMBL7617782 0.73 GAA (0.39) RAB9AKMT2AMEN1ALDH1A1L3MBTL1
SCHEMBL3634188 0.72 ALDH1A1 (0.80) RAB9AKMT2AMEN1ALDH1A1CYP2C9
SCHEMBL16350948 0.72 RAB9A (0.67) RAB9AKMT2AMEN1ALDH1A1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0739903-B1 CARBAMOYLMETHYLUREA DERIVATIVE SHIONOGI & CO (JP) 2002-01-23 EP disclosed
US-5739162-A ANTAGONIST FOR GASTRIN AND/OR CHOLECYSTOKININ B-NOT A-RECEPTORS; SIDE EFFECT REDUCTION; ANTIULCER AGENTS; OPIOD-ENHANCING ANALGESICS; GASTROINTESTINAL DISORDERS; ANXIOLYTIC AGENTS SHIONOGI & CO., LTD. (JP) 1998-04-14 US disclosed
EP-0739903-A1 CARBAMOYLMETHYLUREA DERIVATIVE SHIONOGI & CO., LTD. (JP) 1996-10-30 EP disclosed