SCHEMBL7611075

SCHEMBL7611075

CC(=O)Oc1cc(Cl)ccc1C(=O)NCc1cc(C(F)(F)F)cc(C(F)(F)F)c1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX1 P51575 2/20 0.64
TMPRSS4 Q9NRS4 2/20 0.64
HPGD P15428 2/20 0.53
LMNA P02545 1/20 0.53
MLYCD O95822 1/20 0.47
CYP2C19 P33261 2/20 0.47
KDM4E B2RXH2 1/20 0.47
USP2 O75604 1/20 0.47
ALDH1A1 P00352 1/20 0.47
HSD17B10 Q99714 1/20 0.47
AKR1B1 P15121 3/20 0.46
CCR1 P32246 2/20 0.45
MEN1 O00255 1/20 0.45
PLA2G1B P04054 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
GAA P10253 1/20 0.45
CYP2D6 P10635 1/20 0.45
KMT2A Q03164 1/20 0.45
TDP1 Q9NUW8 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7059962 0.83 AKR1B1 (0.67) P2RX1TMPRSS4HPGDLMNAMLYCD
SCHEMBL13812674 0.78 TMPRSS4 (1.00) P2RX1TMPRSS4HPGDLMNAMLYCD
SCHEMBL7066268 0.78 AKR1B1 (0.62) P2RX1TMPRSS4HPGDLMNAAKR1B1
SCHEMBL3281999 0.74 RHOC (0.56) P2RX1TMPRSS4CYP2C19MEN1CYP1A2
SCHEMBL7063092 0.74 AKR1B1 (0.67) HPGDLMNACYP2C19AKR1B1CCR1
SCHEMBL130511 0.73 TMPRSS4 (0.65) P2RX1TMPRSS4CYP2C19ALDH1A1MEN1
SCHEMBL16088678 0.73 P2RX1 (0.57) P2RX1TMPRSS4HPGDLMNAMLYCD
SCHEMBL13812913 0.72 TMPRSS4 (0.86) P2RX1TMPRSS4HPGDLMNACYP2C19
SCHEMBL16128007 0.71 P2RX1 (0.55) P2RX1TMPRSS4HPGDLMNAMLYCD
SCHEMBL5943436 0.71 ALDH1A1 (0.60) HPGDCYP2C19KDM4EUSP2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1198451-A2 SUBSTITUTED PHENOXYACETIC ACIDS The Institutes for Pharmaceutical Discovery, LLC (US) 2002-04-24 EP disclosed
WO-2001000566-A2 SUBSTITUTED PHENOXYACETIC ACIDS THE INSTITUTES FOR PHARMACEUTICAL DISCOVERY, LLC (US) 2001-01-04 WO disclosed