Bromide

Bromide

SCHEMBL7619356

O=C1[C@H]([P+](c2ccccc2)(c2ccccc2)c2ccccc2)CCN1c1nnc(C(F)(F)F)s1.[Br-]

nearest known ligand 0.45

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHECHKACHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNB1CHRNDCHRNECHRNGHRH2OPRM1

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
OPRM1 known ✓ P35372 1/20 0.41
HTT P42858 3/20 0.45
ALDH1A1 P00352 1/20 0.45
OPRL1 P41146 1/20 0.41
ATM Q13315 1/20 0.37
SLC6A9 P48067 9/20 0.35
HRH3 Q9Y5N1 1/20 0.33
PKM P14618 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
SCD O00767 1/20 0.32
LMNA P02545 1/20 0.31
TSHR P16473 1/20 0.31
HSD17B10 Q99714 1/20 0.31
PARG Q86W56 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL7619352 1.00 HTT (0.45) HTTALDH1A1OPRM1OPRL1ATM
Bromide SCHEMBL8900703 0.76 KMT2A (0.38) ALDH1A1HRH3L3MBTL1KMT2AHSD17B10
Bromide SCHEMBL8558814 0.76 KMT2A (0.38) ALDH1A1HRH3L3MBTL1KMT2AHSD17B10
Bromide SCHEMBL7614674 0.75 L3MBTL1 (0.46) ALDH1A1PKML3MBTL1SCDHSD17B10
Bromide SCHEMBL7614677 0.75 L3MBTL1 (0.46) ALDH1A1PKML3MBTL1SCDHSD17B10
Bromide SCHEMBL8564796 0.74 ALDH1A1 (0.36) HTTALDH1A1KMT2ALMNATSHR
Bromide SCHEMBL8564801 0.74 ALDH1A1 (0.36) HTTALDH1A1KMT2ALMNATSHR
Bromide SCHEMBL7880295 0.73 MEN1 (0.43) MEN1KMT2A
Bromide SCHEMBL7880298 0.73 MEN1 (0.43) MEN1KMT2A
SCHEMBL8788663 0.72 LCAT (0.40) HTTALDH1A1OPRM1OPRL1ATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0620225-B1 Cephalosporin derivatives BASILEA PHARMACEUTICA AG (CH) 2002-11-13 EP disclosed
US-5523400-A 3-(PYRROLIDIN-3-YLIDENE=CH-),7-((2-AMINOTHIAZOL-4-YL)HYDROX -IMINOACETYLAMINO-)-3-CEPHEM DERIVATIVES; BROAD SPECTRUM ANTIBIOTICS HOFFMANN-LA ROCHE INC. (US) 1996-06-04 US disclosed
EP-0620225-A1 Cephalosporin derivatives F. HOFFMANN-LA ROCHE AG (CH) 1994-10-19 EP disclosed