Volkensiflavone

Volkensiflavone

SCHEMBL7620161

O=C1c2c(O)cc(O)cc2OC(c2ccc(O)cc2)C1c1c(O)cc(O)c2c(=O)cc(-c3ccc(O)cc3)oc12

nearest known ligand 0.89

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRSS1 P07477 4/20 0.89
PRSS2 P07478 4/20 0.89
PRSS3 P35030 4/20 0.89
CBS P35520 4/20 0.72
PTPN1 P18031 2/20 0.57
CDK5 Q00535 2/20 0.57
CDK5R1 Q15078 2/20 0.57
BACE1 P56817 2/20 0.56
KLK1 P06870 1/20 0.54
KLK3 P07288 1/20 0.54
KLK2 P20151 1/20 0.54
KLK7 P49862 1/20 0.54
KLK6 Q92876 1/20 0.54
KLK5 Q9Y337 1/20 0.54
PARP1 P09874 2/20 0.52
PARP2 Q9UGN5 1/20 0.52
MMP2 P08253 1/20 0.51
MMP3 P08254 1/20 0.51
MMP9 P14780 1/20 0.51
CYP1A2 P05177 2/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Volkensiflavone SCHEMBL27160551 1.00 PRSS1 (0.89) PRSS1PRSS2PRSS3CBSPTPN1
Volkensiflavone SCHEMBL13829450 1.00 PRSS1 (0.89) PRSS1PRSS2PRSS3CBSPTPN1
SCHEMBL27165462 0.94 PRSS1 (0.90) PRSS1PRSS2PRSS3CBSPTPN1
Morelloflavone SCHEMBL615093 0.94 PRSS1 (1.00) PRSS1PRSS2PRSS3CBSPTPN1
Morelloflavone SCHEMBL2383075 0.94 PRSS1 (1.00) PRSS1PRSS2PRSS3CBSPTPN1
Pancibiflavonol SCHEMBL13829454 0.82 PRSS1 (0.76) PRSS1PRSS2PRSS3CBSPTPN1
SCHEMBL30209479 0.81 PRSS1 (0.62) PRSS1PRSS2PRSS3CBSCYP1A2
SCHEMBL6360019 0.74 KLK1 (0.66) PRSS1PRSS2PRSS3CBSKLK1
SCHEMBL28770111 0.74 KLK1 (0.66) PRSS1PRSS2PRSS3CBSKLK1
SCHEMBL6363033 0.74 KLK1 (0.66) PRSS1PRSS2PRSS3CBSKLK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1245230-A2 Amentoflavone as an antiviral agent Advanced Life Sciences Inc. (US) 2002-10-02 EP disclosed
US-20020068757-A1 Biflavanoids and derivatives thereof as antiviral agents ADVANCED LIFE SCIENCES, INC. 2002-06-06 US disclosed
US-6399654-B1 ADMINISTERING MIXTURE OF VIRICIDE AND BIOFLAVANOID ADVANCED LIFE SCIENCES, INC. 2002-06-04 US disclosed
US-5948918-A PLANT EXTRACTS MEDICHEM RESEARCH, INC. (US) 1999-09-07 US disclosed
WO-1998046238-A1 BIFLAVINOIDS AND DERIVATIVES THEREOF AS ANTIVIRAL AGENTS, ALONE OR IN COMBINATION WITH AT LEAST ONE KNOWN ANTIVIRAL AGENT MEDICHEM RESEARCH, INC. (US) 1998-10-22 WO disclosed
US-5773462-A INFLUENZA THERAPY MEDICHEM RESEARCH, INC. (US) 1998-06-30 US disclosed
EP-0833631-A1 BIFLAVANOIDS AND DERIVATIVES THEREOF AS ANTIVIRAL AGENTS MEDICHEM RESEARCH, INC. (US) 1998-04-08 EP disclosed
WO-1997000679-A1 BIFLAVANOIDS AND DERIVATIVES THEREOF AS ANTIVIRAL AGENTS MEDICHEM RESEARCH, INC. (US) 1997-01-09 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020068757-A1 Biflavanoids and derivatives thereof as antiviral agents HK2, GYS2, HK1 PRSS1 2331/4885PRSS2 1604/4885PRSS3 2085/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.