Morelloflavone

Morelloflavone

SCHEMBL615093

O=C1c2c(O)cc(O)cc2OC(c2ccc(O)cc2)C1c1c(O)cc(O)c2c(=O)cc(-c3ccc(O)c(O)c3)oc12

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRSS1 P07477 4/20 1.00
PRSS2 P07478 4/20 1.00
PRSS3 P35030 4/20 1.00
CBS P35520 2/20 0.73
KLK1 P06870 1/20 0.57
KLK3 P07288 1/20 0.57
KLK2 P20151 1/20 0.57
KLK7 P49862 1/20 0.57
KLK6 Q92876 1/20 0.57
KLK5 Q9Y337 1/20 0.57
PARP1 P09874 3/20 0.53
PARP2 Q9UGN5 2/20 0.53
BACE1 P56817 2/20 0.53
CDK5 Q00535 2/20 0.50
CDK5R1 Q15078 2/20 0.50
PTPN1 P18031 1/20 0.50
KDM4E B2RXH2 3/20 0.49
MEN1 O00255 3/20 0.49
POLB P06746 3/20 0.49
GAA P10253 3/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Morelloflavone SCHEMBL2383075 1.00 PRSS1 (1.00) PRSS1PRSS2PRSS3CBSKLK1
SCHEMBL27165462 0.94 PRSS1 (0.90) PRSS1PRSS2PRSS3CBSKLK1
Volkensiflavone SCHEMBL13829450 0.94 PRSS1 (0.89) PRSS1PRSS2PRSS3CBSKLK1
Volkensiflavone SCHEMBL27160551 0.94 PRSS1 (0.89) PRSS1PRSS2PRSS3CBSKLK1
Volkensiflavone SCHEMBL7620161 0.94 PRSS1 (0.89) PRSS1PRSS2PRSS3CBSKLK1
Pancibiflavonol SCHEMBL13829454 0.86 PRSS1 (0.76) PRSS1PRSS2PRSS3CBSKLK1
SCHEMBL30209479 0.77 PRSS1 (0.62) PRSS1PRSS2PRSS3CBSKDM4E
SCHEMBL16263265 0.74 KLK1 (0.72) PRSS1PRSS2PRSS3CBSKLK1
SCHEMBL6360284 0.74 KLK1 (0.72) PRSS1PRSS2PRSS3CBSKLK1
SCHEMBL29414343 0.74 KLK1 (0.72) PRSS1PRSS2PRSS3CBSKLK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 165 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109010409-A The extraction and purification process and detection method of content of flavonoid compound in a kind of people face fruit leaf 中南民族大学 2018-12-18 CN claimed
CN-106822513-A It is a kind of to treat pharmaceutical composition of osteoproliferation and preparation method thereof 济南昊雨青田医药技术有限公司 2017-06-13 CN claimed
CN-106620064-A Medicinal composition for treating undifferentiated arthritis and preparation method of medicinal composition 济南昊雨青田医药技术有限公司 2017-05-10 CN claimed
CN-106138563-A A kind of pharmaceutical composition treating bladder cancer 济南星懿医药技术有限公司 2016-11-23 CN claimed
CN-105726978-A Summer-heat removing liquid for strengthening infants and preparation method thereof 杭州华威药业股份有限公司 2016-07-06 CN claimed
CN-105596415-A Pharmaceutical composition for treating angina pectoris in coronary heart disease and preparation method thereof JINAN XINGYI MED TECH CO LTD 2016-05-25 CN claimed
CN-105497114-A Pharmaceutical composition for treating dyspepsia and preparation method thereof JINAN XINGYI MED TECH CO LTD 2016-04-20 CN claimed
CN-105288202-A Pharmaceutical composition for curing infantile cough JINAN XINGYI MED TECH CO LTD 2016-02-03 CN claimed
CN-105287739-A Medicine composition for treating leucoderma and preparation method thereof JINAN XINGYI MED TECH CO LTD 2016-02-03 CN claimed
CN-105267289-A Pharmaceutical composition for treating functional dyspepsia and preparation method of pharmaceutical composition JINAN XINGYI MED TECH CO LTD 2016-01-27 CN claimed
US-20120039796-A1 Novel method for creating, suspending and stabilizing electronically modified oxygen derivatives, along with creating, suspending and stabilizing electronically modified reaction intermediates, in a bio compatible fluorocarbon suspension, for the purpose of inducing a cascading immune response in mammalian patients MARKOU DEMETRIOS (US) 2012-02-16 US claimed
US-20110217293-A1 Uses of morelloflavone BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM, THE 2011-09-08 US claimed
WO-2010014199-A2 USES OF MORELLOFLAVONE THE BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2010-02-04 WO claimed
WO-2009023803-A2 MODULATED RELEASE FORMULATION FOR THE DELIVERY OF ONE OR MORE MEDICAMENTS ABBOTT RESPIRATORY LLC (US) 2009-02-19 WO claimed
CN-101049301-A Pharmaceutical preparation of biflavone compound for anti gout HUIBEI COLLEGE OF CHINESE MEDI (CN) 2007-10-10 CN claimed
US-20020068757-A1 Biflavanoids and derivatives thereof as antiviral agents ADVANCED LIFE SCIENCES, INC. 2002-06-06 US claimed
US-6399654-B1 ADMINISTERING MIXTURE OF VIRICIDE AND BIOFLAVANOID ADVANCED LIFE SCIENCES, INC. 2002-06-04 US claimed
WO-1998046238-A1 BIFLAVINOIDS AND DERIVATIVES THEREOF AS ANTIVIRAL AGENTS, ALONE OR IN COMBINATION WITH AT LEAST ONE KNOWN ANTIVIRAL AGENT MEDICHEM RESEARCH, INC. (US) 1998-10-22 WO claimed
EP-0833631-A1 BIFLAVANOIDS AND DERIVATIVES THEREOF AS ANTIVIRAL AGENTS MEDICHEM RESEARCH, INC. (US) 1998-04-08 EP claimed
WO-1997000679-A1 BIFLAVANOIDS AND DERIVATIVES THEREOF AS ANTIVIRAL AGENTS MEDICHEM RESEARCH, INC. (US) 1997-01-09 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020068757-A1 Biflavanoids and derivatives thereof as antiviral agents HK2, GYS2, HK1 PRSS1 2331/4885PRSS2 1604/4885PRSS3 2085/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.