SCHEMBL7623748

SCHEMBL7623748

O=C1C(Cc2ccc(-c3ccccc3)cc2)NC(c2ccc(C(F)(F)F)cc2)=CN1O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.47
GLO1 Q04760 1/20 0.42
KIF11 P52732 2/20 0.41
ROCK2 O75116 1/20 0.38
FFAR1 O14842 1/20 0.38
ACLY P53396 1/20 0.38
GAA P10253 3/20 0.37
BACE1 P56817 1/20 0.37
HDAC1 Q13547 3/20 0.37
HDAC6 Q9UBN7 3/20 0.37
HDAC8 Q9BY41 2/20 0.37
POLB P06746 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C19 P33261 1/20 0.36
LTB4R Q15722 1/20 0.36
LTB4R2 Q9NPC1 1/20 0.36
NPSR1 Q6W5P4 1/20 0.35
PLA2G10 O15496 1/20 0.35
PLA2G5 P39877 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7620532 0.95 CES2 (0.43) CES2GLO1KIF11GAAHDAC1
SCHEMBL7615634 0.91 GAA (0.43) ROCK2GAAHDAC1HDAC6HDAC8
SCHEMBL7622610 0.91 GAA (0.43) ROCK2GAAHDAC1HDAC6HDAC8
SCHEMBL7616025 0.88 GAA (0.45) CES2ROCK2GAAHDAC1HDAC6
SCHEMBL7616794 0.87 NPSR1 (0.45) CES2ROCK2GAAHDAC1HDAC6
SCHEMBL7625943 0.85 GAA (0.47) CES2GAAHDAC1HDAC6HDAC8
SCHEMBL7616578 0.85 ALDH1A1 (0.47) CES2ROCK2GAAPOLBCYP1A2
SCHEMBL7591446 0.85 CES2 (0.44) CES2ROCK2GAAHDAC1HDAC6
SCHEMBL7619044 0.82 NPSR1 (0.49) CES2GAAHDAC1HDAC6HDAC8
SCHEMBL7625933 0.81 GAA (0.50) GAAHDAC1HDAC6HDAC8POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6436933-B1 1-HYDROXY-3-(2-METHYLPROPYL)-5,6-DIPHENYLHYDROPYRAZIN-2-ONE STRUCTURAL BIOINFORMATICS INC. 2002-08-20 US disclosed