SCHEMBL7623786

SCHEMBL7623786

CC1=C(c2ccccc2)NC(Cc2ccccc2)C(=O)N1O

nearest known ligand 0.53

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PLA2G10 O15496 2/20 0.47
PLA2G5 P39877 2/20 0.47
ALDH1A1 P00352 2/20 0.46
GAA P10253 3/20 0.45
POLB P06746 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2C19 P33261 1/20 0.45
ALOX15 P16050 1/20 0.44
HDAC1 Q13547 2/20 0.43
HDAC6 Q9UBN7 2/20 0.43
CES2 O00748 2/20 0.42
HDAC8 Q9BY41 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7626833 0.96 ROCK2 (0.43) PLA2G10PLA2G5ALDH1A1GAAPOLB
SCHEMBL7624222 0.84 GAA (0.46) PLA2G10PLA2G5ALDH1A1GAAPOLB
SCHEMBL7622885 0.82 ROCK2 (0.43) PLA2G10PLA2G5ALDH1A1GAAPOLB
SCHEMBL20516445 0.79 GAA (0.54) PLA2G10PLA2G5ALDH1A1GAAPOLB
SCHEMBL20516443 0.79 GAA (0.54) PLA2G10PLA2G5ALDH1A1GAAPOLB
SCHEMBL7625943 0.71 GAA (0.47) PLA2G10PLA2G5ALDH1A1GAAPOLB
SCHEMBL7616578 0.70 ALDH1A1 (0.47) PLA2G10PLA2G5ALDH1A1GAAPOLB
SCHEMBL7622610 0.69 GAA (0.43) PLA2G10PLA2G5ALDH1A1GAAPOLB
SCHEMBL7616025 0.69 GAA (0.45) PLA2G10PLA2G5ALDH1A1GAAPOLB
SCHEMBL7615634 0.69 GAA (0.43) PLA2G10PLA2G5ALDH1A1GAAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6436933-B1 1-HYDROXY-3-(2-METHYLPROPYL)-5,6-DIPHENYLHYDROPYRAZIN-2-ONE STRUCTURAL BIOINFORMATICS INC. 2002-08-20 US claimed
US-6436933-B1 1-HYDROXY-3-(2-METHYLPROPYL)-5,6-DIPHENYLHYDROPYRAZIN-2-ONE STRUCTURAL BIOINFORMATICS INC. 2002-08-20 US disclosed