SCHEMBL762565

SCHEMBL762565

CC(C)(C)OC(=O)N1CCC[C@@H](c2nc3ccccc3[nH]2)C1

nearest known ligand 0.61

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HPGDS O60760 2/20 0.57
POLB P06746 2/20 0.57
KDM4E B2RXH2 3/20 0.56
HTR2B P41595 4/20 0.51
MAPK1 P28482 1/20 0.49
PRMT5 O14744 1/20 0.49
PARP1 P09874 1/20 0.49
SMN1; SMN2 Q16637 2/20 0.48
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2D6 P10635 1/20 0.48
CYP2C9 P11712 1/20 0.48
CYP2C19 P33261 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19408169 1.00 HPGDS (0.57) HPGDSPOLBKDM4EHTR2BMAPK1
SCHEMBL739188 1.00 HPGDS (0.57) HPGDSPOLBKDM4EHTR2BMAPK1
SCHEMBL24067409 0.90 HTR2B (0.59) POLBHTR2BSMN1; SMN2
SCHEMBL992227 0.88 HTR2B (0.59) HPGDSPOLBHTR2BSMN1; SMN2
SCHEMBL30496093 0.86 HPGDS (0.57) HPGDSMAPK1PRMT5PARP1SMN1; SMN2
SCHEMBL25363420 0.86 HPGDS (0.57) HPGDSMAPK1PRMT5PARP1SMN1; SMN2
SCHEMBL762502 0.85 HPGDS (0.52) HPGDSPOLBKDM4EMAPK1CYP1A2
SCHEMBL743450 0.84 PTGS1 (0.57) HPGDSKDM4EPRMT5PARP1
SCHEMBL743449 0.84 PTGS1 (0.57) HPGDSKDM4EPRMT5PARP1
SCHEMBL742770 0.84 HTR2B (0.50) POLBKDM4EHTR2BSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed