SCHEMBL762502

SCHEMBL762502

CC(C)(C)OC(=O)N1CCC[C@@H](c2nc3ccc(F)cc3[nH]2)C1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGDS O60760 2/20 0.52
CHEK2 O96017 2/20 0.51
BACE1 P56817 5/20 0.50
BACE2 Q9Y5Z0 3/20 0.50
GRIN2B Q13224 1/20 0.49
MPO P05164 1/20 0.49
MAPK1 P28482 1/20 0.49
LMNA P02545 1/20 0.48
POLB P06746 1/20 0.47
KDM4E B2RXH2 3/20 0.46
BRD3 Q15059 1/20 0.46
MEN1 O00255 1/20 0.46
GAA P10253 1/20 0.46
MAPT P10636 1/20 0.46
KMT2A Q03164 1/20 0.46
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2D6 P10635 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL762565 0.85 HPGDS (0.57) HPGDSMAPK1POLBKDM4ECYP1A2
SCHEMBL19408169 0.85 HPGDS (0.57) HPGDSMAPK1POLBKDM4ECYP1A2
SCHEMBL739188 0.85 HPGDS (0.57) HPGDSMAPK1POLBKDM4ECYP1A2
SCHEMBL741433 0.84 MPO (0.55) GRIN2BMPOMAPK1LMNAPOLB
SCHEMBL19385385 0.83 HPGDS (0.48) HPGDSCHEK2GRIN2BMAPK1LMNA
SCHEMBL1299150 0.81 SMN1; SMN2 (0.52) HPGDSLMNAPOLBKDM4EBRD3
SCHEMBL10292467 0.79 HPGDS (0.50) HPGDSCHEK2GRIN2BMAPK1LMNA
SCHEMBL20444734 0.78 CHEK2 (0.44) CHEK2BACE1BACE2KDM4ECYP2D6
SCHEMBL17097142 0.78 BACE1 (0.45) HPGDSCHEK2BACE1BACE2BRD3
SCHEMBL741851 0.77 PARP1 (0.51) HPGDSPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed