SCHEMBL743450

SCHEMBL743450

Cc1cccc2[nH]c([C@@H]3CCCN(C(=O)OC(C)(C)C)C3)nc12

nearest known ligand 0.57

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 1/20 0.57
PTGS2 P35354 1/20 0.57
PARP1 P09874 12/20 0.53
HPGDS O60760 2/20 0.52
HCRTR1 O43613 1/20 0.47
HCRTR2 O43614 1/20 0.47
KDM4E B2RXH2 1/20 0.46
JAK2 O60674 1/20 0.45
JAK1 P23458 1/20 0.45
PRMT5 O14744 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL743449 1.00 PTGS1 (0.57) PTGS1PTGS2PARP1HPGDSHCRTR1
SCHEMBL762497 0.89 PARP1 (0.52) PTGS1PTGS2PARP1HPGDSHCRTR1
SCHEMBL20029041 0.89 PARP1 (0.52) PTGS1PTGS2PARP1HPGDSHCRTR1
SCHEMBL741851 0.88 PARP1 (0.51) PTGS1PTGS2PARP1HPGDSHCRTR1
SCHEMBL741850 0.88 PARP1 (0.51) PTGS1PTGS2PARP1HPGDSHCRTR1
SCHEMBL19951502 0.87 PARP1 (0.70) PARP1
SCHEMBL739188 0.84 HPGDS (0.57) PARP1HPGDSKDM4EPRMT5
SCHEMBL762565 0.84 HPGDS (0.57) PARP1HPGDSKDM4EPRMT5
SCHEMBL19408169 0.84 HPGDS (0.57) PARP1HPGDSKDM4EPRMT5
SCHEMBL30689172 0.78 PARP1 (0.45) PARP1HCRTR1HCRTR2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed