SCHEMBL762813

SCHEMBL762813

[C-]#[N+]c1cc(C(=O)OC(C)(C)C)sc1S(C)(=O)=O

nearest known ligand 0.33

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.33
LMNA P02545 1/20 0.33
MAPK1 P28482 1/20 0.33
CA2 P00918 2/20 0.32
CA12 O43570 1/20 0.32
CA1 P00915 1/20 0.32
CA9 Q16790 1/20 0.32
CA14 Q9ULX7 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL740930 0.74 NR1H2 (0.38) ALDH1A1LMNAMAPK1CA2CA12
SCHEMBL8549434 0.65 TSHR (0.44) ALDH1A1LMNAMAPK1CA2CA12
SCHEMBL17900428 0.62 NPSR1 (0.41) ALDH1A1LMNAMAPK1CA2CA12
SCHEMBL17900429 0.62 ALDH1A1 (0.37) ALDH1A1LMNAMAPK1CA2CA12
SCHEMBL8498605 0.62 GRM6 (0.40) ALDH1A1MAPK1CA2CA12CA1
SCHEMBL8888381 0.62 LMNA (0.44) ALDH1A1LMNAMAPK1CA2CA1
SCHEMBL2412676 0.61 ALDH1A1 (0.55) ALDH1A1CA2CA12CA1CA9
SCHEMBL8887983 0.60 KDM4E (0.46) ALDH1A1LMNAMAPK1
SCHEMBL4345360 0.60 DAO (0.53) ALDH1A1LMNAMAPK1
SCHEMBL8549436 0.60 DAO (0.48) ALDH1A1LMNAMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138217-B2 Aurora kinase inhibitors; proliferative disorders; anticancer agents; antitumor agents; N-(1-methyl-1-phenylethyl)-3-((4-morpholin-4-ylbenzoyl)amino)-1H-thieno(2,3-c)pyrazole-5-carboxamide NERVIANO MEDICAL SCIENCES S.R.L. (IT) 2012-03-20 US disclosed