SCHEMBL763158

SCHEMBL763158

CCCCn1c([C@@H]2CCCNC2)nc2ccccc21

nearest known ligand 0.68

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 5/20 0.68
CHRM1 P11229 3/20 0.68
OPRM1 P35372 2/20 0.52
OPRD1 P41143 2/20 0.52
OPRK1 P41145 2/20 0.52
OPRL1 P41146 2/20 0.52
KCNH2 Q12809 2/20 0.49
ALDH1A1 P00352 1/20 0.49
LMNA P02545 1/20 0.49
HPGD P15428 1/20 0.49
TDP1 Q9NUW8 1/20 0.49
USP2 O75604 1/20 0.49
POLB P06746 1/20 0.49
TLR8 Q9NR97 1/20 0.49
TAAR1 Q96RJ0 1/20 0.48
TP53 P04637 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL739842 0.88 HRH1 (0.70) HRH1CHRM1OPRM1OPRD1OPRK1
SCHEMBL739843 0.88 HRH1 (0.70) HRH1CHRM1OPRM1OPRD1OPRK1
SCHEMBL762533 0.85 CHRM1 (0.51) HRH1CHRM1OPRM1OPRD1OPRK1
Piperidine SCHEMBL742276 0.85 HRH1 (0.67) HRH1CHRM1OPRM1OPRD1OPRK1
Hydrochloric Acid SCHEMBL29205481 0.84 JAK2 (0.53) HRH1CHRM1ALDH1A1LMNAHPGD
Hydrochloric Acid SCHEMBL30881897 0.84 JAK2 (0.53) HRH1CHRM1ALDH1A1LMNAHPGD
SCHEMBL16760326 0.81 TAAR1 (0.63) HRH1CHRM1OPRM1OPRD1OPRK1
SCHEMBL763181 0.81 TLR8 (0.51) HRH1CHRM1TLR8
SCHEMBL743157 0.80 HRH1 (0.63) HRH1CHRM1OPRM1OPRD1OPRK1
SCHEMBL763593 0.80 HRH1 (0.63) HRH1CHRM1OPRM1OPRD1OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed