SCHEMBL763169

SCHEMBL763169

NC[C@@H](CC(=O)O)Cc1ccc(N)c(Br)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA2D1 P54289 2/20 0.37
CACNB3 P54284 1/20 0.37
CACNA1C Q13936 1/20 0.37
PGR P06401 1/20 0.37
ADRA1A P35348 1/20 0.37
HTR2B P41595 1/20 0.37
CACNA2D2 Q9NY47 1/20 0.37
GABBR2 O75899 4/20 0.35
GABBR1 Q9UBS5 4/20 0.35
ALDH1A1 P00352 1/20 0.35
CDC25B P30305 1/20 0.35
CASP6 P55212 1/20 0.35
RCE1 Q9Y256 1/20 0.35
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA4 P22748 1/20 0.33
CA6 P23280 1/20 0.33
CA5A P35218 1/20 0.33
CA7 P43166 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL763137 0.78 CACNA2D1 (0.43) CACNA2D1CACNB3CACNA1CPGRADRA1A
SCHEMBL16070906 0.75 SLC7A5 (0.58) ADORA3KDM4EUSP2EGFRLCK
SCHEMBL29808980 0.74 GAA (0.50) ALDH1A1CDC25BCASP6RCE1CA2
SCHEMBL4168904 0.74 CPA1 (0.56) CACNA2D1CACNB3CACNA1CPGRADRA1A
SCHEMBL2434720 0.74 GAA (0.50) ALDH1A1CDC25BCASP6RCE1CA2
Hydrochloric Acid SCHEMBL30898977 0.74 SLC7A5 (0.57) ADORA3KDM4EUSP2EGFRLCK
Hydrochloric Acid SCHEMBL30898984 0.74 SLC7A5 (0.57) ADORA3KDM4EUSP2EGFRLCK
SCHEMBL6459207 0.72 LDHA (0.61) ALDH1A1CA12CA1CA2CA5A
SCHEMBL762549 0.72 LOXL2 (0.50) ALDH1A1CA2LMNACYP1A2CYP2C19
Bicarbonate SCHEMBL9288170 0.71 CES2 (0.44) ALDH1A1CDC25BCASP6RCE1CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed