SCHEMBL7635345

SCHEMBL7635345

Oc1ccc(C(CCNCC(O)COc2cccc3[nH]ccc23)c2ccc(O)cc2)cc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 11/20 0.60
ADRB2 P07550 7/20 0.58
ADRB1 P08588 7/20 0.58
ADRB3 P13945 7/20 0.58
CYP1A2 P05177 2/20 0.58
CYP3A4 P08684 2/20 0.58
LMNA P02545 2/20 0.58
KDM4E B2RXH2 1/20 0.58
USP2 O75604 1/20 0.58
CYP2D6 P10635 1/20 0.58
THRB P10828 1/20 0.58
CYP2C9 P11712 1/20 0.58
TSHR P16473 1/20 0.58
TP53 P04637 1/20 0.58
GLA P06280 1/20 0.58
ALOX15 P16050 1/20 0.58
NFKB1 P19838 1/20 0.58
DRD4 P21917 1/20 0.58
HTR1B P28222 1/20 0.58
HTR2C P28335 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7641388 0.90 HTR1A (0.61) HTR1AADRB2ADRB1ADRB3CYP1A2
SCHEMBL6322237 0.89 ADRB3 (0.65) HTR1AADRB2ADRB1ADRB3CYP1A2
SCHEMBL6056296 0.81 HTR1A (0.71) HTR1AADRB2ADRB1ADRB3CYP1A2
SCHEMBL7296138 0.81 ADRB3 (0.78) ADRB2ADRB1ADRB3
SCHEMBL7288262 0.79 ADRB3 (0.69) HTR1AADRB2ADRB1ADRB3CYP1A2
SCHEMBL7297780 0.78 ADRB3 (0.68) HTR1AADRB2ADRB1ADRB3CYP1A2
SCHEMBL4845543 0.78 HTR1A (0.76) HTR1AADRB2ADRB1ADRB3CYP1A2
SCHEMBL7367227 0.78 HTR1A (0.61) HTR1AADRB2ADRB1ADRB3CYP1A2
SCHEMBL7296273 0.77 ADRB3 (0.67) HTR1AADRB2ADRB1ADRB3CYP1A2
SCHEMBL7285328 0.77 ADRB3 (0.67) HTR1AADRB2ADRB1ADRB3CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1230210-A1 AMINOALCOHOL DERIVATIVES USEFUL FOR THE TREATMENT OF GASTROINTESTINAL DISORDERS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2002-08-14 EP disclosed
WO-2001036375-A1 AMINOALCOHOL DERIVATIVES USEFUL FOR THE TREATMENT OF GASTROINTESTINAL DISORDERS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-05-25 WO disclosed