SCHEMBL7636710

SCHEMBL7636710

CC(=O)OCC1C(=O)N2C(C(=O)O)=CCS[C@@H]12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1I2 O75469 3/20 0.39
PGR P06401 2/20 0.39
PTGS2 P35354 2/20 0.39
TDP1 Q9NUW8 4/20 0.39
KDM4E B2RXH2 2/20 0.39
TSHR P16473 1/20 0.39
HSD17B10 Q99714 1/20 0.39
MAPT P10636 3/20 0.37
ALDH1A1 P00352 1/20 0.37
CYP3A4 P08684 1/20 0.37
APEX1 P27695 1/20 0.37
SLC15A2 Q16348 1/20 0.37
SPOP O43791 1/20 0.36
PTGS1 P23219 1/20 0.34
L3MBTL1 Q9Y468 3/20 0.33
ESR1 P03372 1/20 0.33
KDR P35968 1/20 0.33
HPGD P15428 1/20 0.32
DNMT1 P26358 1/20 0.32
SLC22A6 Q4U2R8 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8077885 0.87 NR1I2 (0.42) NR1I2PGRPTGS2TDP1KDM4E
SCHEMBL9388602 0.86 NR1I2 (0.38) NR1I2PGRPTGS2TDP1KDM4E
SCHEMBL10693978 0.86 NR1I2 (0.39) NR1I2PGRPTGS2TDP1KDM4E
SCHEMBL10436335 0.82 KDM4E (0.40) NR1I2PGRPTGS2TDP1KDM4E
SCHEMBL9198941 0.81 SPOP (0.41) NR1I2PGRPTGS2TDP1KDM4E
SCHEMBL9190737 0.81 KDM4E (0.41) NR1I2PGRPTGS2TDP1KDM4E
SCHEMBL10670083 0.80 KDM4E (0.42) NR1I2PGRPTGS2TDP1KDM4E
SCHEMBL10582215 0.76 MAPT (0.40) NR1I2PGRPTGS2TDP1KDM4E
SCHEMBL9295936 0.75 KDM4E (0.34) NR1I2PGRPTGS2TDP1KDM4E
SCHEMBL6066202 0.75 NR1I2 (0.42) NR1I2PGRPTGS2TDP1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0230972-A2 Method of producing cephem compounds Takeda Chemical Industries, Ltd. (JP) 1987-08-05 EP claimed
US-6458948-B1 MIXING A QUATERNARY AMMONIUM SALT HAVING A PARTICULAR TRIAZINE RING IN THE MOLECULES THEREOF, A CARBOXYLIC ACID COMPOUND AND A COMPOUND HAVING A NUCLEOPHILIC FUNCTIONAL GROUP, TO CONDENSE THE CARBOXYLIC ACID WITH THE COMPOUND HAVING THE NUCLEOPHILIC TOKUYAMA CORPORATION (JP) 2002-10-01 US disclosed
EP-0251299-A2 Cephalosporin compounds, processes for their preparation and antibacterial agents Kaken Pharmaceutical Co., Ltd. (JP) 1988-01-07 EP disclosed
EP-0091130-A2 Cephalosporin derivatives, process for preparing and pharmaceutical compositions containing said compounds DAIICHI SEIYAKU CO., LTD. (JP) 1983-10-12 EP disclosed