SCHEMBL763705

SCHEMBL763705

CCCCn1c([C@@H]2CCCN(C(=O)C[C@H](N)Cc3ccc(-c4ccc5c(c4)OCCN5C)cc3)C2)nc2c(F)cccc21

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SYK P43405 1/20 0.34
KDM1A O60341 2/20 0.34
HDAC4 P56524 1/20 0.34
HRH1 P35367 3/20 0.33
MDM2 Q00987 1/20 0.33
CYP2D6 P10635 2/20 0.33
PDCD1 Q15116 1/20 0.33
CD274 Q9NZQ7 1/20 0.33
GRM5 P41594 1/20 0.33
CFD P00746 2/20 0.33
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
METAP2 P50579 1/20 0.32
CYP11B1 P15538 1/20 0.32
CYP11B2 P19099 1/20 0.32
DPP4 P27487 2/20 0.31
PIK3CD O00329 1/20 0.31
PIK3CB P42338 1/20 0.31
DGAT1 O75907 1/20 0.31
DPP8 Q6V1X1 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL740111 0.93 CFD (0.34) SYKKDM1AHDAC4HRH1MDM2
SCHEMBL740110 0.93 CFD (0.34) SYKKDM1AHDAC4HRH1MDM2
SCHEMBL739093 0.85 CFD (0.35) HRH1CYP2D6PDCD1CD274CFD
SCHEMBL739094 0.85 CFD (0.35) HRH1CYP2D6PDCD1CD274CFD
SCHEMBL741729 0.84 SYK (0.35) SYKHDAC4HRH1MDM2PDCD1
SCHEMBL741728 0.84 SYK (0.35) SYKHDAC4HRH1MDM2PDCD1
SCHEMBL742755 0.83 HRH1 (0.39) HDAC4HRH1CYP2D6PIK3CDPIK3CB
SCHEMBL742754 0.83 HRH1 (0.39) HDAC4HRH1CYP2D6PIK3CDPIK3CB
SCHEMBL741288 0.82 CFD (0.36) HRH1CYP2D6CFDDPP4DPP8
SCHEMBL741289 0.82 CFD (0.36) HRH1CYP2D6CFDDPP4DPP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed