SCHEMBL763813

SCHEMBL763813

COCCCn1c([C@@H]2CCCN(C(=O)C[C@@H](Cc3ccc4ccccc4c3)NC(=O)OC(C)(C)C)C2)nc2c1CCCC2

nearest known ligand 0.37

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CTSB P07858 1/20 0.37
CTSS P25774 1/20 0.37
CTSK P43235 1/20 0.37
PADI4 Q9UM07 2/20 0.35
KLK5 Q9Y337 1/20 0.35
PPIA P62937 2/20 0.35
HRH2 P25021 1/20 0.34
HRH1 P35367 1/20 0.34
GHSR Q92847 1/20 0.34
ACE P12821 1/20 0.33
SCN9A Q15858 1/20 0.33
MCHR1 Q99705 2/20 0.32
PPARA Q07869 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL762785 0.89 HRH1 (0.42) CTSBCTSSCTSKPADI4HRH1
SCHEMBL763304 0.87 ALDH1A1 (0.35) HRH1PPARA
SCHEMBL762648 0.86 HRH1 (0.36) CTSBCTSSCTSKPADI4KLK5
SCHEMBL763816 0.86 CTSB (0.36) CTSBCTSSCTSKPADI4KLK5
SCHEMBL10293031 0.86 PADI4 (0.38) CTSBCTSSCTSKPADI4KLK5
SCHEMBL762559 0.86 KCNH2 (0.39) CTSBCTSSCTSKPADI4KLK5
SCHEMBL763177 0.86 CTSB (0.36) CTSBCTSSCTSKPADI4KLK5
SCHEMBL10292140 0.86 PADI4 (0.37) CTSBCTSSCTSKPADI4KLK5
SCHEMBL762577 0.86 CTSB (0.36) CTSBCTSSCTSKPADI4KLK5
SCHEMBL740450 0.86 ALDH1A1 (0.35) HRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed