SCHEMBL763304

SCHEMBL763304

COCCCn1c([C@@H]2CCCN(C(=O)C[C@H](C)Cc3ccc4ccccc4c3)C2)nc2c1CCCC2

nearest known ligand 0.36

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.35
TSHR P16473 3/20 0.35
KMT2A Q03164 2/20 0.35
KCNH2 Q12809 2/20 0.35
CYP2D6 P10635 2/20 0.35
HRH1 P35367 2/20 0.35
BCHE P06276 4/20 0.34
LMNA P02545 2/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
PPARA Q07869 1/20 0.34
HTT P42858 1/20 0.34
RAB9A P51151 1/20 0.34
POLB P06746 1/20 0.34
CNR2 P34972 1/20 0.33
MEN1 O00255 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL740450 0.92 ALDH1A1 (0.35) ALDH1A1TSHRKMT2AKCNH2CYP2D6
SCHEMBL740451 0.92 ALDH1A1 (0.35) ALDH1A1TSHRKMT2AKCNH2CYP2D6
SCHEMBL763813 0.87 CTSB (0.37) HRH1PPARA
SCHEMBL742676 0.87 CYP2D6 (0.34) ALDH1A1TSHRKMT2AKCNH2CYP2D6
SCHEMBL762546 0.84 KCNH2 (0.37) ALDH1A1TSHRKMT2AKCNH2CYP2D6
SCHEMBL762548 0.84 KCNH2 (0.40) ALDH1A1TSHRKMT2AKCNH2CYP2D6
SCHEMBL739244 0.79 HRH1 (0.46) KCNH2CYP2D6HRH1POLB
SCHEMBL739245 0.79 HRH1 (0.46) KCNH2CYP2D6HRH1POLB
SCHEMBL741263 0.78 KCNH2 (0.38) KMT2AKCNH2CYP2D6HRH1
SCHEMBL740883 0.78 KCNH2 (0.38) KMT2AKCNH2CYP2D6HRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed