SCHEMBL764236

SCHEMBL764236

O=C(c1ccc(-c2cccs2)cc1)N1CCCC1

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 4/20 0.76
BCR P11274 4/20 0.76
HPGD P15428 6/20 0.61
MAPK1 P28482 1/20 0.61
ALDH1A1 P00352 3/20 0.58
GAA P10253 1/20 0.57
SLC6A2 P23975 1/20 0.54
SLC6A4 P31645 1/20 0.54
SLC6A3 Q01959 1/20 0.54
NPC1 O15118 2/20 0.53
RAB9A P51151 2/20 0.53
TP53 P04637 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
HDAC3 O15379 2/20 0.52
HDAC1 Q13547 2/20 0.52
HDAC2 Q92769 2/20 0.52
PKM P14618 1/20 0.51
ADORA2A P29274 2/20 0.51
TACR3 P29371 1/20 0.50
MEN1 O00255 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10198116 0.97 ABL1 (0.76) ABL1BCRHPGDMAPK1ALDH1A1
SCHEMBL27556543 0.87 ABL1 (0.71) ABL1BCRHPGDMAPK1ALDH1A1
SCHEMBL911426 0.79 ABL1 (0.64) ABL1BCRALDH1A1TACR3
SCHEMBL4052776 0.78 ABL1 (0.50) ABL1BCRHPGDALDH1A1GAA
SCHEMBL764268 0.77 ABL1 (0.54) ABL1BCRHPGDALDH1A1GAA
SCHEMBL764282 0.77 HDAC3 (0.52) ABL1BCRHPGDALDH1A1GAA
SCHEMBL10721733 0.77 HPGD (0.95) HPGDMAPK1ALDH1A1MEN1TSHR
SCHEMBL3901121 0.76 HDAC3 (0.62) ABL1BCRHPGDALDH1A1GAA
SCHEMBL764280 0.76 ABL1 (0.53) ABL1BCRHPGDALDH1A1GAA
SCHEMBL6614562 0.76 HPGD (1.00) HPGDMAPK1ALDH1A1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2078015-B1 MODULATORS OF GLUCOCORTICOID RECEPTOR, AP-1 AND/OR NF-KAPPAB ACTIVITY AND USE THEREOF BRISTOL MYERS SQUIBB CO (US) 2012-03-21 EP disclosed