SCHEMBL764282

SCHEMBL764282

O=C(c1ccc(-c2cccs2)cc1Cl)N1CCCC1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 3/20 0.52
HDAC1 Q13547 3/20 0.52
HDAC2 Q92769 3/20 0.52
HPGD P15428 3/20 0.50
NPC1 O15118 1/20 0.50
ALDH1A1 P00352 1/20 0.50
TP53 P04637 1/20 0.50
RAB9A P51151 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
ABL1 P00519 4/20 0.49
BCR P11274 4/20 0.49
GAA P10253 1/20 0.49
KDM4E B2RXH2 1/20 0.47
USP2 O75604 1/20 0.46
KCNH2 Q12809 1/20 0.45
HRH3 Q9Y5N1 1/20 0.45
KMT2A Q03164 1/20 0.45
POLB P06746 1/20 0.44
TSHR P16473 1/20 0.44
GRIN2B Q13224 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL764268 0.84 ABL1 (0.54) HDAC3HDAC1HDAC2HPGDNPC1
SCHEMBL3901121 0.83 HDAC3 (0.62) HDAC3HDAC1HDAC2HPGDNPC1
SCHEMBL764280 0.83 ABL1 (0.53) HDAC3HDAC1HDAC2HPGDNPC1
SCHEMBL3901114 0.82 HDAC3 (0.55) HDAC3HDAC1HDAC2HPGDNPC1
SCHEMBL10331354 0.79 YEATS4 (0.54) HDAC3HDAC1HDAC2HPGDNPC1
SCHEMBL764236 0.77 ABL1 (0.76) HDAC3HDAC1HDAC2HPGDNPC1
SCHEMBL10331952 0.75 HPGD (0.53) HPGDNPC1ALDH1A1RAB9ASMN1; SMN2
SCHEMBL10198116 0.75 ABL1 (0.76) HDAC3HDAC1HDAC2HPGDNPC1
SCHEMBL24508969 0.74 P2RX7 (0.60) HPGDNPC1TP53RAB9ASMN1; SMN2
SCHEMBL29944105 0.72 MEN1 (0.62) HPGDNPC1TP53RAB9AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2078015-B1 MODULATORS OF GLUCOCORTICOID RECEPTOR, AP-1 AND/OR NF-KAPPAB ACTIVITY AND USE THEREOF BRISTOL MYERS SQUIBB CO (US) 2012-03-21 EP disclosed