SCHEMBL7646115

SCHEMBL7646115

CCCOCC(=O)c1ccc(I)cc1

nearest known ligand 0.53

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 2/20 0.44
TPMT P51580 1/20 0.41
ALDH1A1 P00352 2/20 0.40
SLC6A2 P23975 2/20 0.40
ESR1 P03372 1/20 0.40
CHRM1 P11229 1/20 0.40
TSHR P16473 1/20 0.40
KDR P35968 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
CA1 P00915 2/20 0.39
CA2 P00918 2/20 0.39
HSD17B3 P37058 1/20 0.39
SLC6A4 P31645 1/20 0.38
SLC6A3 Q01959 1/20 0.38
PDPK1 O15530 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11461527 0.84 PLA2G4B (0.50) L3MBTL1ALDH1A1TSHR
SCHEMBL862846 0.84 HSD17B3 (0.58) ALDH1A1SLC6A2ESR1CHRM1TSHR
SCHEMBL7650212 0.82 L3MBTL1 (0.44) L3MBTL1ALDH1A1SLC6A2ESR1CHRM1
SCHEMBL2126591 0.81 LMNA (0.56) L3MBTL1ALDH1A1TDP1
SCHEMBL8218440 0.81 L3MBTL1 (0.68) L3MBTL1ALDH1A1TSHR
SCHEMBL7646419 0.81 HDAC3 (0.56) L3MBTL1ALDH1A1
SCHEMBL7646664 0.79 HAO1 (0.46) L3MBTL1ALDH1A1SLC6A2ESR1CHRM1
SCHEMBL6963661 0.77 SMN1; SMN2 (0.54) L3MBTL1ALDH1A1TDP1
SCHEMBL6040897 0.77 TPMT (0.46) TPMTCA1CA2PDPK1
SCHEMBL11444536 0.77 GSK3B (0.54) L3MBTL1ALDH1A1TSHRTDP1CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6479520-B1 REGULATING APOPTOSIS IN HUMAN CELLS WITH COMPOUNDS SUCH AS: 3-CYANO-6-(2-METHOXY-4-METHYLTHIOIPHENYL)-2(1H)-PYRIDINONE CELL PATHWAYS, INC. 2002-11-12 US disclosed
US-6046216-A USEFUL TO INHIBIT THE GROWTH OF NEOPLASTIC CELLS. CELL PATHWAYS, INC. (US) 2000-04-04 US disclosed
EP-0428268-A2 Pharmaceutical phenylpyridone derivatives SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1991-05-22 EP disclosed