SCHEMBL7649207

SCHEMBL7649207

CCCCC1=NN(Cc2ccc(-c3ccccc3C#N)cc2)C(CCCC)N1

nearest known ligand 0.47

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ACHE P22303 2/20 0.47
PPARG P37231 2/20 0.46
AGTR1 P30556 5/20 0.44
AGTR2 P50052 2/20 0.40
LTB4R2 Q9NPC1 2/20 0.39
PRKAG1 P54619 3/20 0.38
PRKAA1 Q13131 3/20 0.38
PRKAB1 Q9Y478 3/20 0.38
CNR2 P34972 1/20 0.38
APLNR P35414 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2692039 0.74 PPARG (0.53) ACHEPPARGAGTR1AGTR2
SCHEMBL9402468 0.73 ACHE (0.44) ACHEPPARGAGTR1AGTR2LTB4R2
SCHEMBL5411252 0.72 AGTR1 (0.43) ACHEPPARGAGTR1AGTR2LTB4R2
SCHEMBL4253889 0.70 HSD17B10 (0.58) ACHEPPARGAGTR1AGTR2
SCHEMBL9402217 0.69 POLB (0.66) ACHEPPARGAGTR1AGTR2
SCHEMBL1894100 0.69 AGTR1 (0.68) ACHEPPARGAGTR1AGTR2
SCHEMBL9682387 0.69 AGTR1 (0.43) ACHEPPARGAGTR1AGTR2LTB4R2
SCHEMBL6954317 0.69 HSD17B10 (0.60) ACHEPPARGAGTR1AGTR2
SCHEMBL10718048 0.69 HSD17B10 (0.60) ACHEPPARGAGTR1AGTR2
SCHEMBL6954649 0.69 HSD17B10 (0.60) ACHEPPARGAGTR1AGTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6358984-B1 FOR THERAPY OF HYPERTENSION AND/OR DISEASES SUCH AS HEART AND RENAL DISEASES LEAD CHEMICAL CO., LTD. (JP) 2002-03-19 US disclosed
US-6232335-B1 A BIPHENYL TRIAZOLE COMPOUND USEFUL AS A ANGIOTENSIN II CONVERTING ENZYME INHIBITORS EFFECTIVE IN THE TREATMENT OF HYPERTENSION OR HEART FAILURE LEAD CHEMICAL CO., LTD. (JP) 2001-05-15 US disclosed