SCHEMBL7650358

SCHEMBL7650358

CC1=C(NNC(=O)OCc2ccccc2)[CH]CC=C1

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.49
RAB9A P51151 1/20 0.49
P2RX7 Q99572 1/20 0.45
GAA P10253 1/20 0.43
CA12 O43570 2/20 0.43
CA1 P00915 2/20 0.43
CA2 P00918 2/20 0.43
CA9 Q16790 2/20 0.43
POLB P06746 1/20 0.43
ALDH1A1 P00352 1/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
MAOB P27338 1/20 0.42
LMNA P02545 1/20 0.42
MGLL Q99685 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6991431 0.76 NPC1 (0.51) NPC1RAB9AGAACA12CA1
SCHEMBL7654986 0.75 P2RX7 (0.48) NPC1RAB9AP2RX7GAACA12
SCHEMBL2295789 0.72 CA12 (0.66) NPC1RAB9AP2RX7GAACA12
SCHEMBL4908338 0.71 GAA (0.69) NPC1RAB9AP2RX7GAACA12
SCHEMBL2918702 0.71 GAA (0.64) NPC1RAB9AP2RX7GAACA12
SCHEMBL27880557 0.70 CA12 (0.60) NPC1RAB9AP2RX7GAACA12
SCHEMBL4149248 0.69 ALDH1A1 (0.60) NPC1RAB9AP2RX7CA12CA1
Hydrochloric Acid SCHEMBL4149246 0.68 ALDH1A1 (0.58) NPC1RAB9AP2RX7CA12CA1
SCHEMBL28954497 0.68 ALDH1A1 (0.63) NPC1RAB9AP2RX7CA12CA1
SCHEMBL11651843 0.67 CA12 (0.60) NPC1RAB9AP2RX7CA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6462076-B2 CYSTEINE PROTEASE INHIBITORS USEFUL FOR THE TREATMENT OF DISEASES ASSOCIATED WITH CYSTEINE PROTEASES, SUCH AS OSTEOPOROSIS, OSTEOARTHRITIS, RHEUMATOID ARTHRITIS, TUMOR METASTASIS, ANGINA PECTORIS, PLAQUE RUPTURE AND STROKE ETC. HOFFMANN-LA ROCHE INC. 2002-10-08 US disclosed