SCHEMBL765151

SCHEMBL765151

CC1CC(c2nc3ccccc3[nH]2)CN(C(=O)C[C@@H](Cc2ccc3ccccc3c2)NC(=O)OC(C)(C)C)C1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 1/20 0.41
CTSB P07858 1/20 0.40
CTSS P25774 1/20 0.40
CTSK P43235 1/20 0.40
GHSR Q92847 1/20 0.37
CXCR3 P49682 1/20 0.36
POLB P06746 3/20 0.36
MAPT P10636 1/20 0.36
ITGB3 P05106 1/20 0.36
ITGAV P06756 1/20 0.36
HTR2B P41595 1/20 0.36
BDKRB2 P30411 1/20 0.36
KDM4E B2RXH2 3/20 0.36
BCHE P06276 1/20 0.36
KMT2A Q03164 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.35
MAPK1 P28482 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL762987 0.84 HTR2B (0.42) CXCR3POLBMAPTHTR2BKDM4E
SCHEMBL762864 0.82 MAPK1 (0.45) CTSBCTSSCTSKPOLBMAPT
SCHEMBL762586 0.82 CYP1A2 (0.42) CTSBCTSSCTSKPOLBKDM4E
SCHEMBL741088 0.81 HTR2B (0.39) CXCR3POLBHTR2BKDM4EKMT2A
SCHEMBL762654 0.81 MAPK1 (0.43) CTSBCTSSCTSKPOLBMAPT
SCHEMBL763211 0.81 CYP1A2 (0.41) CTSBCTSSCTSKPOLBKDM4E
SCHEMBL763789 0.80 CTSB (0.37) CTSBCTSSCTSKPOLBMAPT
SCHEMBL763468 0.80 GRIN2B (0.49) PTPN1POLBMAPTITGB3ITGAV
SCHEMBL763367 0.80 GRIN2B (0.49) PTPN1POLBMAPTITGB3ITGAV
SCHEMBL762470 0.80 GRIN2B (0.49) PTPN1POLBMAPTITGB3ITGAV

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed