SCHEMBL765163

SCHEMBL765163

COC(=O)N1CCc2c([nH]c3ccc(Cl)cc23)C1c1ccc(C)cc1

nearest known ligand 0.55

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TP53 P04637 6/20 0.55
MAPT P10636 4/20 0.55
SMN1; SMN2 Q16637 1/20 0.55
ABCG2 Q9UNQ0 2/20 0.55
KIF11 P52732 7/20 0.54
LMNA P02545 2/20 0.54
SIRT1 Q96EB6 1/20 0.54
HTR2A P28223 2/20 0.53
HTR2C P28335 2/20 0.53
POLB P06746 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL764793 0.95 TP53 (0.58) TP53MAPTSMN1; SMN2ABCG2KIF11
SCHEMBL11912895 0.92 KIF11 (0.59) TP53MAPTSMN1; SMN2ABCG2KIF11
SCHEMBL9961950 0.92 KIF11 (0.63) TP53MAPTABCG2KIF11LMNA
SCHEMBL9961949 0.92 KIF11 (0.63) TP53MAPTABCG2KIF11LMNA
SCHEMBL8402724 0.91 KIF11 (0.55) TP53MAPTSMN1; SMN2ABCG2KIF11
SCHEMBL763913 0.91 ABCG2 (0.60) TP53MAPTSMN1; SMN2ABCG2KIF11
SCHEMBL764923 0.91 TP53 (0.66) TP53MAPTSMN1; SMN2ABCG2KIF11
SCHEMBL764584 0.91 TP53 (0.67) TP53MAPTSMN1; SMN2ABCG2KIF11
SCHEMBL8402733 0.91 KIF11 (0.60) TP53MAPTSMN1; SMN2ABCG2KIF11
SCHEMBL765206 0.90 KIF11 (0.57) TP53MAPTSMN1; SMN2ABCG2KIF11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 65 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080103164-A1 USEFUL COMPOUNDS FOR HPV INFECTION SMITHKLINE BEECHAM CORPORATION 2008-05-01 US claimed
EP-1786425-A1 USEFUL COMPOUNDS FOR HPV INFECTION SmithKline Beecham Corporation (US) 2007-05-23 EP claimed
WO-2007002051-A1 CARBOLINE DERIVATIVES AND THEIR USE AS INHIBITORS OF FLAVIVIRIDAE INFECTIONS SMITHKLINE BEECHAM CORPORATION (US) 2007-01-04 WO claimed
WO-2006015035-A1 USEFUL COMPOUNDS FOR HPV INFECTION SMITHKLINE BEECHAM CORPORATION (US) 2006-02-09 WO claimed
US-20240043422-A1 METHODS FOR TREATING CANCER AND NON-NEOPLASTIC CONDITIONS PTC THERAPEUTICS, INC. (US) 2024-02-08 US disclosed
US-11613538-B2 Method of inhibiting or reducing a viral infection PTC THERAPEUTICS, INC. (US) 2023-03-28 US disclosed
EP-2434891-B9 METHODS FOR TREATING CANCER AND NON-NEOPLASTIC CONDITIONS PTC THERAPEUTICS INC (US) 2021-05-05 EP disclosed
US-20200317668-A1 METHOD OF INHIBITING OR REDUCING A CORONAVIRIDAE VIRUS INFECTION PTC THERAPEUTICS, INC. 2020-10-08 US disclosed
EP-3718405-A1 METHODS FOR TREATING CANCER AND NON-NEOPLASTIC CONDITIONS PTC Therapeutics, Inc. (US) 2020-10-07 EP disclosed
EP-2434891-B1 METHODS FOR TREATING CANCER AND NON-NEOPLASTIC CONDITIONS PTC THERAPEUTICS INC (US) 2020-07-22 EP disclosed
US-20190194188-A1 METHODS FOR TREATING CANCER AND NON-NEOPLASTIC CONDITIONS PTC THERAPEUTICS, INC. 2019-06-27 US disclosed
US-20160340354-A1 METHODS FOR TREATING CANCER AND NON-NEOPLASTIC CONDITIONS PTC THERAPEUTICS, INC. 2016-11-24 US disclosed
US-20070281962-A2 Administering 1,2,3,6-tetrasubstituted pyrido[3,4-b]indoles to inhibit the 5'-untranslated region-dependent translation; anticarcinogenic agents; retinopathy, rheumatoid arthritis, psoriasis, atherosclerosis, obesity, macular degeneration PCT THERAPEUTICS, INC. (US) 2007-12-06 US disclosed
US-20070281962-A2 Administering 1,2,3,6-tetrasubstituted pyrido[3,4-b]indoles to inhibit the 5'-untranslated region-dependent translation; anticarcinogenic agents; retinopathy, rheumatoid arthritis, psoriasis, atherosclerosis, obesity, macular degeneration PCT THERAPEUTICS, INC. (US) 2007-12-06 US disclosed
US-20070254878-A1 ADMINISTRATION OF CARBOLINE DERIVATIVES USEFUL IN THE TREATMENT OF CANCER AND OTHER DISEASES PTC THERAPEUTICS, INC. 2007-11-01 US disclosed
US-20070254878-A1 ADMINISTRATION OF CARBOLINE DERIVATIVES USEFUL IN THE TREATMENT OF CANCER AND OTHER DISEASES PTC THERAPEUTICS, INC. 2007-11-01 US disclosed
WO-2005089764-A9 CARBOLINE DERIVATIVES USEFUL IN THE INHIBITION OF ANGIOGENESIS PTC THERAPEUTICS INC (US) 2007-09-13 WO disclosed
EP-1786425-A1 USEFUL COMPOUNDS FOR HPV INFECTION SmithKline Beecham Corporation (US) 2007-05-23 EP disclosed
WO-2007002051-A1 CARBOLINE DERIVATIVES AND THEIR USE AS INHIBITORS OF FLAVIVIRIDAE INFECTIONS SMITHKLINE BEECHAM CORPORATION (US) 2007-01-04 WO disclosed
WO-2006015035-A1 USEFUL COMPOUNDS FOR HPV INFECTION SMITHKLINE BEECHAM CORPORATION (US) 2006-02-09 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240043422-A1 METHODS FOR TREATING CANCER AND NON-NEOPLASTIC CONDITIONS HDGF, POLRMT, VEGFA TP53 15/4885MAPT 3300/4885SMN1; SMN2 3502/4885
US-20160340354-A1 METHODS FOR TREATING CANCER AND NON-NEOPLASTIC CONDITIONS HDGF, POLRMT, VEGFA TP53 16/4885MAPT 3328/4885SMN1; SMN2 3473/4885
US-20190194188-A1 METHODS FOR TREATING CANCER AND NON-NEOPLASTIC CONDITIONS HDGF, POLRMT, VEGFA TP53 16/4885MAPT 3328/4885SMN1; SMN2 3473/4885
US-20070254878-A1 ADMINISTRATION OF CARBOLINE DERIVATIVES USEFUL IN THE TREATMENT OF CANCER AND OTHER DISEASES VEGFA, FLT4, FLT1 TP53 52/4885MAPT 3997/4885SMN1; SMN2 3261/4885
US-20200317668-A1 METHOD OF INHIBITING OR REDUCING A CORONAVIRIDAE VIRUS INFECTION SARS1, POLRMT, EIF2AK2 TP53 1818/4885MAPT 2964/4885SMN1; SMN2 4373/4885
US-11613538-B2 Method of inhibiting or reducing a viral infection SARS1, EIF2AK2, POLRMT TP53 1710/4885MAPT 2901/4885SMN1; SMN2 4142/4885
US-20080103164-A1 USEFUL COMPOUNDS FOR HPV INFECTION TP53, POLI, PCNA TP53 1/4885MAPT 4453/4885SMN1; SMN2 4792/4885
US-20070281962-A2 Administering 1,2,3,6-tetrasubstituted pyrido[3,4-b]indoles to inhibit the 5'-untranslated region-dependent translation; anticarcinogenic agents; retinopathy, rheumatoid arthritis, psoriasis, atherosclerosis, obesity, macular degeneration VEGFA, FLT4, MIF TP53 448/4885MAPT 2854/4885SMN1; SMN2 4645/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.