SCHEMBL7651780

SCHEMBL7651780

Cc1ccc2c(ccc3c(C(F)(F)F)nn(-c4ccc(S(N)(=O)=O)cc4)c32)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 14/20 0.54
PTGS1 P23219 11/20 0.54
PDPK1 O15530 5/20 0.54
PTGES O14684 2/20 0.54
HDAC3 O15379 1/20 0.54
CA12 O43570 1/20 0.54
PDE5A O76074 1/20 0.54
ABCB11 O95342 1/20 0.54
MT-CO2 P00403 1/20 0.54
CA1 P00915 1/20 0.54
CA2 P00918 1/20 0.54
LMNA P02545 1/20 0.54
CA3 P07451 1/20 0.54
CYP3A4 P08684 1/20 0.54
ALOX5 P09917 1/20 0.54
ADORA3 P0DMS8 1/20 0.54
CYP2D6 P10635 1/20 0.54
CYP2C9 P11712 1/20 0.54
ADRB3 P13945 1/20 0.54
ALOX15 P16050 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8917761 0.89 PTGS2 (0.53) PTGS2PTGS1CYP2D6CYP2C9
SCHEMBL9229049 0.87 PTGS2 (0.55) PTGS2PTGS1PDPK1
SCHEMBL9233734 0.87 PTGS2 (0.57) PTGS2PTGS1PDPK1CA1CA2
SCHEMBL9233871 0.86 PDPK1 (0.60) PTGS2PTGS1PDPK1CA12CA1
SCHEMBL8917361 0.85 PTGS2 (0.56) PTGS2PTGS1PDPK1CA12CA1
SCHEMBL7649968 0.85 PTGS2 (0.53) PTGS2PTGS1PDPK1PTGESHDAC3
SCHEMBL8918086 0.83 PTGS2 (0.48) PTGS2PTGS1PDPK1CA12CA1
SCHEMBL8917480 0.82 PTGS2 (0.49) PTGS2PTGS1PDPK1
SCHEMBL9235959 0.81 PTGS2 (0.53) PTGS2PTGS1PDPK1PTGESHDAC3
SCHEMBL8917853 0.79 PTGS2 (0.52) PTGS2PTGS1CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6492411-B1 TREATING ARTHRITIS; REDUCED SIDE EFFECTS G. D. SEARLE & CO. 2002-12-10 US disclosed