SCHEMBL7652187

SCHEMBL7652187

Cc1ccc2[nH]cc(C(C)NC3=CC(=O)c4cccnc4C3=O)c2c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NQO1 P15559 2/20 0.49
TDP2 O95551 2/20 0.48
G6PD P11413 2/20 0.48
NSD2 O96028 2/20 0.48
CDC25B P30305 1/20 0.48
DUSP3 P51452 1/20 0.48
HKDC1 Q2TB90 1/20 0.48
S100A4 P26447 2/20 0.44
MAPT P10636 6/20 0.38
TP53 P04637 4/20 0.38
SMN1; SMN2 Q16637 3/20 0.37
TGM2 P21980 1/20 0.37
PADI1 Q9ULC6 1/20 0.37
PADI3 Q9ULW8 1/20 0.37
PADI4 Q9UM07 1/20 0.37
PADI2 Q9Y2J8 1/20 0.37
RAB9A P51151 2/20 0.35
GSK3A P49840 1/20 0.34
GSK3B P49841 1/20 0.34
GUSB P08236 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7647844 0.89 NQO1 (0.48) NQO1TDP2G6PDNSD2CDC25B
SCHEMBL7652382 0.89 TDP2 (0.49) NQO1TDP2G6PDNSD2CDC25B
SCHEMBL7679049 0.88 NQO1 (0.60) NQO1TDP2G6PDNSD2CDC25B
SCHEMBL7648036 0.88 NQO1 (0.47) NQO1TDP2G6PDNSD2CDC25B
SCHEMBL15698456 0.78 NQO1 (0.76) NQO1TDP2G6PDNSD2S100A4
SCHEMBL7647843 0.73 TDP2 (0.58) NQO1TDP2G6PDNSD2CDC25B
SCHEMBL7648029 0.73 TDP2 (0.58) NQO1TDP2G6PDNSD2CDC25B
SCHEMBL7648160 0.73 TDP2 (0.74) NQO1TDP2G6PDNSD2CDC25B
SCHEMBL7678312 0.70 TDP2 (0.60) NQO1TDP2G6PDNSD2CDC25B
SCHEMBL7654680 0.70 CDC25B (0.60) NQO1TDP2G6PDNSD2CDC25B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012064396-A9 NOVEL EZRIN INHIBITORS AND METHODS OF MAKING AND USING GEORGETOWN UNIVERSITY (US) 2012-07-05 WO disclosed
WO-2012064396-A2 NOVEL EZRIN INHIBITORS AND METHODS OF MAKING AND USING GEORGETOWN UNIVERSITY (US) 2012-05-18 WO disclosed