SCHEMBL7652383

SCHEMBL7652383

CC(O)C(N1CCN(Cc2ccc(C(C)(C)C)cc2)CC1)n1c2ccccc2c2ccccc21

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 4/20 0.50
NR1I2 O75469 1/20 0.50
ADORA3 P0DMS8 1/20 0.50
CNR1 P21554 1/20 0.50
HRH1 P35367 1/20 0.50
OPRK1 P41145 1/20 0.50
PDE4D Q08499 1/20 0.50
KCNH2 Q12809 1/20 0.50
GHSR Q92847 1/20 0.50
GAA P10253 1/20 0.46
OPRD1 P41143 1/20 0.46
MAPK1 P28482 2/20 0.46
HTT P42858 2/20 0.46
MEN1 O00255 3/20 0.45
KMT2A Q03164 3/20 0.45
MAPT P10636 3/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
DNM1 Q05193 1/20 0.42
TP53 P04637 4/20 0.41
DRD2 P14416 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7647493 0.92 MAPT (0.49) LMNANR1I2ADORA3CNR1HRH1
SCHEMBL7649700 0.88 LMNA (0.59) LMNAGAAMAPK1HTTMEN1
SCHEMBL7649894 0.86 MEN1 (0.49) LMNAGAAMAPK1HTTMEN1
SCHEMBL7648593 0.86 GPR183 (0.44) LMNANR1I2ADORA3CNR1HRH1
SCHEMBL7646684 0.84 MAPT (0.48) LMNAKCNH2GAAMAPK1HTT
SCHEMBL7653466 0.84 LMNA (0.65) LMNAGAAMAPK1HTTMEN1
SCHEMBL7650388 0.82 CHKA (0.41) MEN1KMT2AMAPTSMN1; SMN2TP53
SCHEMBL7649923 0.81 ALDH1A1 (0.49) LMNAMAPK1MEN1KMT2AMAPT
SCHEMBL7653796 0.80 MAPT (0.50) LMNAGAAMAPK1HTTMEN1
SCHEMBL7651629 0.80 LMNA (0.50) LMNAGAAOPRD1MAPK1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1237887-A1 9-(PIPERAZINYLALKYL)CARBAZOLES AS BAX-MODULATORS Applied Research Systems ARS Holding N.V. (AN) 2002-09-11 EP disclosed
WO-2001029028-A1 9- (PIPERAZINYLALKYL) CARBAZOLES AS BAX-MODULATORS APPLIED RESEARCH SYSTEMS ARS HOLDING N.V. (AN) 2001-04-26 WO disclosed