SCHEMBL7652999

SCHEMBL7652999

O=C(O)[C@H](CNCc1ccc(N2CCN(c3ncccn3)CC2)cc1)NS(=O)(=O)c1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 9/20 0.52
ITGA2B P08514 9/20 0.52
ALDH1A1 P00352 2/20 0.46
MDM2 Q00987 1/20 0.46
ITGAV P06756 2/20 0.46
CA1 P00915 2/20 0.46
CA2 P00918 2/20 0.46
CA7 P43166 2/20 0.46
CA9 Q16790 2/20 0.46
TSHR P16473 1/20 0.43
MAPK1 P28482 1/20 0.43
LMNA P02545 1/20 0.42
MAPT P10636 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
MMP2 P08253 1/20 0.41
MMP13 P45452 1/20 0.41
SLC6A7 Q99884 1/20 0.41
MMP3 P08254 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL381814 0.85 ITGB3 (0.55) ITGB3ITGA2BALDH1A1ITGAVTSHR
SCHEMBL7654405 0.84 ITGB3 (0.74) ITGB3ITGA2BITGAV
SCHEMBL7649709 0.83 ITGB3 (0.56) ITGB3ITGA2BITGAV
SCHEMBL7651226 0.83 ITGB3 (0.46) ITGB3ITGA2BALDH1A1MDM2ITGAV
SCHEMBL7653684 0.82 ITGB3 (0.70) ITGB3ITGA2BITGAV
SCHEMBL7653489 0.82 ITGB3 (0.46) ITGB3ITGA2BALDH1A1ITGAVLMNA
SCHEMBL7653020 0.80 ALDH1A1 (0.43) ITGB3ITGA2BALDH1A1MDM2CA1
SCHEMBL6496630 0.78 ITGB3 (0.59) ITGB3ITGA2BITGAV
SCHEMBL7651973 0.78 ITGB3 (0.54) ITGB3ITGA2BITGAVLMNASMN1; SMN2
SCHEMBL7651943 0.78 ITGB3 (0.60) ITGB3ITGA2BITGAV

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6451800-B1 Phenylpiperazine derivatives as integrin αvβ3 antagonists MEIJI SEIKA KAISHA, LTD. (JP) 2002-09-17 US claimed
EP-1057818-A1 PHENYLPIPERAZINE DERIVATIVES AS INTEGRIN ALPHAvBETA3 ANTAGONISTS MEIJI SEIKA KAISHA LTD. (JP) 2000-12-06 EP claimed
US-6451800-B1 Phenylpiperazine derivatives as integrin αvβ3 antagonists MEIJI SEIKA KAISHA, LTD. (JP) 2002-09-17 US disclosed
EP-1057818-A1 PHENYLPIPERAZINE DERIVATIVES AS INTEGRIN ALPHAvBETA3 ANTAGONISTS MEIJI SEIKA KAISHA LTD. (JP) 2000-12-06 EP disclosed