SCHEMBL765300

SCHEMBL765300

COC(=O)C(Cc1ccc(C)cc1)NC=O

nearest known ligand 0.54

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ATM Q13315 2/20 0.54
L3MBTL1 Q9Y468 1/20 0.54
NOS2 P35228 2/20 0.45
NOS3 P29474 1/20 0.45
NOS1 P29475 1/20 0.45
ALDH1A1 P00352 1/20 0.43
THRB P10828 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
HSD17B10 Q99714 1/20 0.43
HDAC1 Q13547 4/20 0.42
HDAC6 Q9UBN7 4/20 0.42
ESR1 P03372 1/20 0.42
ESR2 Q92731 1/20 0.42
POLB P06746 1/20 0.42
KMT2A Q03164 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
TSHR P16473 1/20 0.40
LNPEP Q9UIQ6 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29057553 0.88 ESR1 (0.56) ATMNOS2NOS3NOS1ALDH1A1
SCHEMBL10587222 0.88 ESR1 (0.56) ATMNOS2NOS3NOS1ALDH1A1
SCHEMBL22804064 0.88 ESR1 (0.56) ATMNOS2NOS3NOS1ALDH1A1
SCHEMBL1503825 0.86 NOS2 (0.54) ATML3MBTL1NOS2NOS3NOS1
SCHEMBL6658615 0.86 NOS2 (0.44) ATML3MBTL1NOS2NOS3NOS1
SCHEMBL11549702 0.86 LNPEP (0.45) ATML3MBTL1NOS2NOS3NOS1
SCHEMBL6572040 0.86 LNPEP (0.45) ATML3MBTL1NOS2NOS3NOS1
SCHEMBL3499885 0.86 ATM (0.58) ATML3MBTL1NOS2NOS3NOS1
SCHEMBL27925079 0.86 ATM (0.58) ATML3MBTL1NOS2NOS3NOS1
SCHEMBL1274700 0.86 ATM (0.58) ATML3MBTL1NOS2NOS3NOS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1577301-B1 Antithrombotic diaminocyclohexane derivatives DAIICHI SANKYO CO LTD (JP) 2012-09-12 EP disclosed
EP-1270557-B1 ETHYLENEDIAMINE DERIVATIVES DAIICHI SANKYO CO LTD (JP) 2012-07-25 EP disclosed
EP-2431370-A1 Monoacylated 1,2-diaminocycloalkanes DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2012-03-21 EP disclosed