SCHEMBL7653540

SCHEMBL7653540

Nc1nc(Cl)cc(NCc2ccc(C(=O)O)cc2)n1

nearest known ligand 0.70

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.53
SMN1; SMN2 Q16637 2/20 0.53
CYP2D6 P10635 1/20 0.51
CYP2C19 P33261 1/20 0.51
HRH4 Q9H3N8 2/20 0.47
L3MBTL1 Q9Y468 2/20 0.44
KMT2A Q03164 2/20 0.44
MEN1 O00255 1/20 0.44
EPHX2 P34913 1/20 0.44
PTGS2 P35354 3/20 0.44
VCP P55072 1/20 0.43
PTGES O14684 1/20 0.43
ALOX5 P09917 1/20 0.43
POLB P06746 1/20 0.43
HPGD P15428 1/20 0.43
HSD17B10 Q99714 1/20 0.43
CTDSP1 Q9GZU7 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17315168 0.87 ALDH1A1 (0.72) ALDH1A1SMN1; SMN2CYP2D6CYP2C19HRH4
SCHEMBL1319082 0.83 SMN1; SMN2 (0.68) ALDH1A1SMN1; SMN2CYP2D6CYP2C19HRH4
SCHEMBL7655249 0.82 SMN1; SMN2 (0.46) ALDH1A1SMN1; SMN2CYP2D6CYP2C19HRH4
SCHEMBL18177427 0.81 HRH4 (0.63) ALDH1A1SMN1; SMN2CYP2D6CYP2C19HRH4
SCHEMBL23291905 0.78 ALDH1A1 (0.49) ALDH1A1CYP2D6CYP2C19L3MBTL1KMT2A
SCHEMBL5251108 0.78 CYP2D6 (0.51) ALDH1A1SMN1; SMN2CYP2D6CYP2C19HRH4
SCHEMBL18177442 0.77 SMN1; SMN2 (0.53) ALDH1A1SMN1; SMN2CYP2D6CYP2C19HRH4
SCHEMBL17315282 0.76 ALDH1A1 (0.72) ALDH1A1SMN1; SMN2CYP2D6CYP2C19HRH4
SCHEMBL443320 0.76 HCAR2 (0.55) ALDH1A1SMN1; SMN2L3MBTL1KMT2AMEN1
SCHEMBL13322077 0.73 SMN1; SMN2 (0.46) ALDH1A1SMN1; SMN2CYP2D6CYP2C19HRH4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6489333-B2 HETEROCYCLIC COMPOUNDS CONTAINING A GUANIDINE MIMIC, FOR INHIBITION OF CELL ADHESION, TREATMENT OF ANGIOGENESIS DISORDERS, INFLAMMATION, CANCER METASTASIS, DIABETIC RETINOPATHY, THROMBOSIS, RESTENOSIS, MACULAR DEGENERATION BRISTOL - MEYERS SQUIBB PHARMA COMPANY 2002-12-03 US disclosed
US-20010044535-A1 Integrin antagonists BRISTOL-MYERS SQUIBB PHARMA COMPANY 2001-11-22 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20010044535-A1 Integrin antagonists ITGB3, VCAM1, ITGB2 ALDH1A1 2216/4885SMN1; SMN2 2789/4885CYP2D6 2646/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.