SCHEMBL7653696

SCHEMBL7653696

C=C(C)C1c2cc(NC(=O)c3ccc(OCC)c(Br)c3)ccc2CCN1C

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 13/20 0.61
SMN1; SMN2 Q16637 6/20 0.61
HSD17B10 Q99714 2/20 0.61
ALOX15 P16050 1/20 0.61
ALOX12 P18054 1/20 0.61
NR4A1 P22736 1/20 0.61
MEN1 O00255 6/20 0.53
KMT2A Q03164 6/20 0.53
TP53 P04637 5/20 0.53
KDM4E B2RXH2 3/20 0.48
HTT P42858 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
NPC1 O15118 1/20 0.48
MAPK1 P28482 1/20 0.48
LMNA P02545 3/20 0.45
POLB P06746 3/20 0.45
ALDH1A1 P00352 2/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2C9 P11712 1/20 0.45
HPGD P15428 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7993838 0.87 MAPT (0.65) MAPTSMN1; SMN2HSD17B10ALOX15ALOX12
SCHEMBL7655483 0.87 MAPT (0.43) MAPTSMN1; SMN2HSD17B10ALOX15ALOX12
SCHEMBL7008578 0.80 MAPT (0.56) MAPTSMN1; SMN2HSD17B10ALOX15ALOX12
SCHEMBL6293914 0.80 MAPT (0.68) MAPTSMN1; SMN2HSD17B10ALOX15ALOX12
SCHEMBL7012423 0.80 MAPT (0.55) MAPTSMN1; SMN2HSD17B10ALOX15ALOX12
SCHEMBL7661456 0.79 RORC (0.47) MAPTSMN1; SMN2HSD17B10MEN1KMT2A
SCHEMBL7657907 0.79 MAPT (0.63) MAPTSMN1; SMN2HSD17B10ALOX15ALOX12
SCHEMBL7652942 0.79 MAPT (0.47) MAPTSMN1; SMN2MEN1KMT2ATP53
SCHEMBL7658675 0.77 ROCK2 (0.42) TP53LMNA
SCHEMBL6294927 0.77 MAPT (0.61) MAPTSMN1; SMN2HSD17B10ALOX15ALOX12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6492378-B1 Substituted isoquinoline derivatives and their use as anticonvulsivants SMITHKLINE BEECHAM P.L.C. (GB) 2002-12-10 US disclosed