SCHEMBL7658675

SCHEMBL7658675

C=C(C)C1c2cc(NC(=O)c3ccc(OC(C)C)c(C#N)c3)ccc2CCN1C

nearest known ligand 0.50

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 5/20 0.42
S1PR1 P21453 9/20 0.41
LMNA P02545 1/20 0.40
TP53 P04637 1/20 0.40
NPY2R P49146 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7654464 0.88 ROCK2 (0.41) ROCK2TP53
SCHEMBL7661456 0.87 RORC (0.47) ROCK2LMNATP53
Hydrochloric Acid SCHEMBL6293630 0.82 ROCK2 (0.57) ROCK2S1PR1
SCHEMBL7009661 0.81 RORC (0.49) ROCK2NPY2R
Hydrochloric Acid SCHEMBL7007842 0.80 RORC (0.48) ROCK2NPY2R
SCHEMBL7652942 0.77 MAPT (0.47) ROCK2TP53
SCHEMBL8145389 0.77 ROCK2 (0.53) ROCK2S1PR1TP53
SCHEMBL7653696 0.77 MAPT (0.61) LMNATP53
SCHEMBL7655014 0.76 ALDH1A1 (0.39) ROCK2S1PR1TP53NPY2R
SCHEMBL7655483 0.75 MAPT (0.43) LMNATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6492378-B1 Substituted isoquinoline derivatives and their use as anticonvulsivants SMITHKLINE BEECHAM P.L.C. (GB) 2002-12-10 US disclosed