SCHEMBL7653829

SCHEMBL7653829

CC(=O)On1c(=O)c(-c2cn(CCCN)c3ccc(Br)cc23)nc2cc3c(cc21)CCC3

nearest known ligand 0.36

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 4/20 0.36
CNR1 P21554 3/20 0.36
CAMK2D Q13557 2/20 0.36
DYRK1A Q13627 1/20 0.35
GSK3B P49841 10/20 0.35
QPCT Q16769 8/20 0.33
PDK1 Q15118 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7666393 0.98 CAMK2D (0.36) CNR2CNR1CAMK2DDYRK1AGSK3B
SCHEMBL7662842 0.91 PDE4B (0.40) GSK3BQPCTPDK1
SCHEMBL7665495 0.90 CAMK2D (0.41) CAMK2DGSK3B
SCHEMBL7662560 0.90 PDE4B (0.40) GSK3BQPCT
SCHEMBL7664149 0.89 CAMK2D (0.41) CAMK2DGSK3B
SCHEMBL7663936 0.88 CAMK2D (0.39) CNR2CAMK2DGSK3B
SCHEMBL7841757 0.87 DYRK1A (0.38) CNR2CAMK2DDYRK1AGSK3BQPCT
SCHEMBL7664668 0.86 MAOB (0.40)
SCHEMBL7657124 0.86 CAMK2D (0.39) CNR2CAMK2DGSK3B
SCHEMBL7853098 0.86 KDM4E (0.33) GSK3BQPCT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6458792-B1 MEDICAMENT FOR THE TREATMENT OF INFLAMMATORY, IMMUNOLOGICAL, BRONCHOPULMONARY, CARDIOVASCULAR, ONCOLOGICAL OR CNS-DEGENERATIVE DISORDERS. ASTRAZENECA AB (SE) 2002-10-01 US disclosed
EP-1071683-A1 NEW COMPOUNDS AstraZeneca AB (SE) 2001-01-31 EP disclosed
WO-1999046264-A1 NEW COMPOUNDS ASTRAZENECA AB (SE) 1999-09-16 WO disclosed