SCHEMBL7654510

SCHEMBL7654510

CN1C2CCC1CC(OC(=O)c1cc(Cl)c(Cl)cc1C(=O)OC1CC3CCC(C1)N3C)C2

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 5/20 0.68
HTR3E A5X5Y0 5/20 0.68
HTR3B O95264 5/20 0.68
HTR3A P46098 5/20 0.68
HTR3D Q70Z44 5/20 0.68
HTR3C Q8WXA8 5/20 0.68
CYP1A2 P05177 2/20 0.68
MTOR P42345 2/20 0.68
GMNN O75496 1/20 0.68
ALOX15 P16050 1/20 0.68
TSHR P16473 1/20 0.68
PMP22 Q01453 1/20 0.68
HSD17B10 Q99714 1/20 0.68
GAA P10253 1/20 0.66
CYP2C19 P33261 2/20 0.62
LMNA P02545 2/20 0.62
MEN1 O00255 1/20 0.61
KMT2A Q03164 1/20 0.61
NR1I2 O75469 1/20 0.61
CHRNA7 P36544 2/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7654509 1.00 CYP2D6 (0.68) CYP2D6HTR3EHTR3BHTR3AHTR3D
SCHEMBL10635123 0.85 CYP2D6 (0.66) CYP2D6HTR3EHTR3BHTR3AHTR3D
SCHEMBL6507167 0.84 HTR3E (0.66) CYP2D6HTR3EHTR3BHTR3AHTR3D
SCHEMBL6507170 0.84 HTR3E (0.66) CYP2D6HTR3EHTR3BHTR3AHTR3D
SCHEMBL5789235 0.83 CYP2D6 (0.71) CYP2D6HTR3EHTR3BHTR3AHTR3D
SCHEMBL5789236 0.83 CYP2D6 (0.71) CYP2D6HTR3EHTR3BHTR3AHTR3D
SCHEMBL5787520 0.82 HTR3E (0.59) CYP2D6HTR3EHTR3BHTR3AHTR3D
SCHEMBL7652481 0.81 HTR3A (0.75) CYP2D6HTR3EHTR3BHTR3AHTR3D
SCHEMBL7652475 0.81 HTR3A (0.75) CYP2D6HTR3EHTR3BHTR3AHTR3D
Bemesetron SCHEMBL10765684 0.81 CYP2D6 (1.00) CYP2D6HTR3EHTR3BHTR3AHTR3D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6376510-B1 ADMINISTERING A ALKOXY- AND ACYLOXY-SUBSTITUTED ARALKYL AND ARALKENYL BIS QUATERNARY AMMONIUM DERIVATIVES OF CYCLIC ALKANOL DIESTERS TO A HUMAN AS MUSCLE RELAXANTS NEWLAXANT LLC 2002-04-23 US disclosed
US-6274757-B1 REACTING AN HYDROXY AMINE CORRESPONDING COMPOUND WITH DICHLORO COMPOUND NEWLAXANT LLC 2001-08-14 US disclosed