SCHEMBL7659052

SCHEMBL7659052

CN(C)c1ccc2c(c1)c(=O)[nH]c(=O)n2CCCCN1CCC(OC(c2ccccc2)c2ccccc2)CC1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCHE P06276 10/20 0.46
HPGDS O60760 1/20 0.43
P2RX7 Q99572 4/20 0.43
CHRM2 P08172 3/20 0.43
CHRM1 P11229 3/20 0.43
SLC6A2 P23975 3/20 0.43
ADRA1A P35348 3/20 0.43
DRD3 P35462 3/20 0.43
SLC6A3 Q01959 3/20 0.43
KCNH2 Q12809 3/20 0.43
HTR1A P08908 2/20 0.43
ADRA2A P08913 2/20 0.43
DRD1 P21728 2/20 0.43
MLNR O43193 2/20 0.43
NR1I2 O75469 2/20 0.43
LMNA P02545 2/20 0.43
ADORA3 P0DMS8 2/20 0.43
DRD2 P14416 2/20 0.43
ADRA2C P18825 2/20 0.43
CHRM3 P20309 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7653211 0.94 BCHE (0.46) BCHEHPGDSP2RX7CHRM2CHRM1
SCHEMBL7656321 0.89 BCHE (0.48) BCHEHPGDSP2RX7CHRM2CHRM1
SCHEMBL7651720 0.87 BCHE (0.48) BCHEHPGDSP2RX7CHRM2CHRM1
SCHEMBL7654569 0.87 BCHE (0.53) BCHEHPGDSP2RX7SLC6A2ADRA1A
SCHEMBL7649496 0.86 BCHE (0.53) BCHEHPGDSP2RX7CHRM2CHRM1
SCHEMBL7648364 0.85 P2RX7 (0.53) BCHEHPGDSP2RX7CHRM2CHRM1
SCHEMBL7653124 0.85 BCHE (0.55) BCHEHPGDSP2RX7CHRM2CHRM1
SCHEMBL7654787 0.85 BCHE (0.42) BCHEHPGDSP2RX7CHRM2CHRM1
SCHEMBL7654420 0.84 P2RX7 (0.52) BCHEHPGDSP2RX7CHRM2CHRM1
SCHEMBL7651628 0.84 BCHE (0.52) BCHEHPGDSCHRM2CHRM1SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6407116-B1 2,4-DIOXO-1,2,3,4-TETRAHYDROQUINAZOLINE DERIVATIVES; ANTIALLERGENS, ANTIASTHMATICS, ANTIHISTAMINES, AND ANTIINFLAMMATORY AGENTS TAKEDA CHEMICAL INDUSTRIES, INC. (JP) 2002-06-18 US disclosed
EP-1026160-A1 NITROGENOUS FUSED-RING COMPOUNDS, PROCESS FOR THE PREPARATION OF THE SAME, AND DRUGS Takeda Chemical Industries, Ltd. (JP) 2000-08-09 EP disclosed