SCHEMBL7654639

SCHEMBL7654639

O=C1C=C(O)/C(=C/c2ccccc2-c2ccc(Cn3cncn3)cc2)O1

nearest known ligand 0.42

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 15/20 0.42
HDAC1 Q13547 2/20 0.38
HDAC6 Q9UBN7 2/20 0.38
KDM4E B2RXH2 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7654440 0.77 CYP19A1 (0.56) CYP19A1HDAC1HDAC6
SCHEMBL7657762 0.73 CYP19A1 (0.43) CYP19A1HDAC1HDAC6
SCHEMBL6693307 0.68 CYP19A1 (0.61) CYP19A1HDAC1HDAC6
SCHEMBL6700110 0.67 CYP19A1 (0.56) CYP19A1HDAC1HDAC6
SCHEMBL8304477 0.67 KDM4E (0.32) KDM4E
SCHEMBL7674570 0.67 CYP19A1 (0.79) CYP19A1HDAC1HDAC6KDM4E
SCHEMBL305950 0.67 CYP19A1 (0.63) CYP19A1HDAC1HDAC6
SCHEMBL8305411 0.67 KDM4E (0.31) KDM4E
SCHEMBL15688800 0.66 CYP19A1 (0.71) CYP19A1HDAC1HDAC6
SCHEMBL7655658 0.65 CYP19A1 (0.75) CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6358984-B1 FOR THERAPY OF HYPERTENSION AND/OR DISEASES SUCH AS HEART AND RENAL DISEASES LEAD CHEMICAL CO., LTD. (JP) 2002-03-19 US disclosed
US-6232335-B1 A BIPHENYL TRIAZOLE COMPOUND USEFUL AS A ANGIOTENSIN II CONVERTING ENZYME INHIBITORS EFFECTIVE IN THE TREATMENT OF HYPERTENSION OR HEART FAILURE LEAD CHEMICAL CO., LTD. (JP) 2001-05-15 US disclosed