SCHEMBL8304477

SCHEMBL8304477

CC1=NN(c2ccc(-c3ccccc3/C=C3\OC(=O)C=C3O)cc2)CN1

nearest known ligand 0.32

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2C19 P33261 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8300516 0.75 ACHE (0.31)
SCHEMBL8305411 0.68 KDM4E (0.31) KDM4ECYP1A2CYP2C19
SCHEMBL27406701 0.68 APP (0.44) KDM4ECYP1A2
SCHEMBL7654639 0.67 CYP19A1 (0.42) KDM4E
SCHEMBL8522511 0.67
SCHEMBL8303502 0.66
SCHEMBL8306226 0.64
SCHEMBL7658574 0.64 APLNR (0.32)
SCHEMBL7660666 0.64 BRS3 (0.32)
SCHEMBL8304618 0.64 KDM4E (0.33) KDM4ECYP1A2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0936221-A1 NOVEL 2,4-DIOXOPYRROLIDINE AND 2,4-DIOXOTETRAHYDROFURAN DERIVATIVES AND MEDICINES CONTAINING THE SAME AS THE ACTIVE INGREDIENT LEAD CHEMICAL COMPANY LTD. (JP) 1999-08-18 EP disclosed