SCHEMBL7654998

SCHEMBL7654998

CN(Cc1ccc(N2CCN(C3=NCCCN3)CC2)cc1)C(CC(=O)O)NS(=O)(=O)c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 10/20 0.44
ITGA2B P08514 10/20 0.44
ITGAV P06756 9/20 0.44
RORC P51449 6/20 0.37
ALDH1A1 P00352 2/20 0.37
PKM P14618 1/20 0.37
ITGB1 P05556 1/20 0.37
ITGB5 P18084 1/20 0.37
CNR2 P34972 2/20 0.36
CNR1 P21554 1/20 0.36
RORB Q92753 1/20 0.36
LMNA P02545 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7652576 0.91 ITGB3 (0.45) ITGB3ITGA2BITGAVRORCALDH1A1
SCHEMBL7653506 0.84 NPC1 (0.42) ITGB3ITGA2BRORCALDH1A1PKM
SCHEMBL7654994 0.83 ITGB3 (0.51) ITGB3ITGA2BITGAVITGB1ITGB5
SCHEMBL7649721 0.83 ITGB3 (0.45) ITGB3ITGA2BITGAVALDH1A1PKM
SCHEMBL7653746 0.82 ITGB3 (0.46) ITGB3ITGA2BITGAVALDH1A1PKM
SCHEMBL7652565 0.81 ITGB3 (0.52) ITGB3ITGA2BITGAVRORCITGB1
SCHEMBL7650148 0.80 ITGB3 (0.48) ITGB3ITGA2BITGAVALDH1A1PKM
SCHEMBL7651202 0.80 ITGB3 (0.53) ITGB3ITGA2BITGAVALDH1A1PKM
SCHEMBL7649709 0.78 ITGB3 (0.56) ITGB3ITGA2BITGAVITGB1ITGB5
SCHEMBL7654234 0.77 ITGB3 (0.63) ITGB3ITGA2BITGAVRORCITGB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6451800-B1 Phenylpiperazine derivatives as integrin αvβ3 antagonists MEIJI SEIKA KAISHA, LTD. (JP) 2002-09-17 US claimed
EP-1057818-A1 PHENYLPIPERAZINE DERIVATIVES AS INTEGRIN ALPHAvBETA3 ANTAGONISTS MEIJI SEIKA KAISHA LTD. (JP) 2000-12-06 EP claimed
US-6451800-B1 Phenylpiperazine derivatives as integrin αvβ3 antagonists MEIJI SEIKA KAISHA, LTD. (JP) 2002-09-17 US disclosed
EP-1057818-A1 PHENYLPIPERAZINE DERIVATIVES AS INTEGRIN ALPHAvBETA3 ANTAGONISTS MEIJI SEIKA KAISHA LTD. (JP) 2000-12-06 EP disclosed