SCHEMBL7650148

SCHEMBL7650148

O=C(O)CC(NS(=O)(=O)c1ccccc1)N(CC1CC1)C(=O)c1ccc(N2CCN(C3=NCCCN3)CC2)cc1

nearest known ligand 0.48

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 15/20 0.48
ITGA2B P08514 14/20 0.48
ITGAV P06756 14/20 0.48
ITGB1 P05556 1/20 0.35
ITGB5 P18084 1/20 0.35
LIMK2 P53671 1/20 0.34
HTR2A P28223 1/20 0.33
HTR2C P28335 1/20 0.33
HTR7 P34969 1/20 0.33
ALDH1A1 P00352 1/20 0.33
PKM P14618 1/20 0.33
MMP3 P08254 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7653746 0.88 ITGB3 (0.46) ITGB3ITGA2BITGAVITGB1ITGB5
SCHEMBL383369 0.88 ITGB3 (0.64) ITGB3ITGA2BITGAVITGB1ITGB5
SCHEMBL7653577 0.86 NPC1 (0.41) ITGB3ITGA2BITGAVLIMK2HTR2A
SCHEMBL7650144 0.83 ITGB3 (0.55) ITGB3ITGA2BITGAVITGB1ITGB5
SCHEMBL27475491 0.81 ITGB3 (0.46) ITGB3ITGA2BITGAVLIMK2ALDH1A1
SCHEMBL383511 0.81 ITGB3 (0.46) ITGB3ITGA2BITGAVLIMK2ALDH1A1
SCHEMBL7652576 0.81 ITGB3 (0.45) ITGB3ITGA2BITGAVITGB1ITGB5
SCHEMBL7654998 0.80 ITGB3 (0.44) ITGB3ITGA2BITGAVITGB1ITGB5
SCHEMBL7651202 0.80 ITGB3 (0.53) ITGB3ITGA2BITGAVITGB1ITGB5
SCHEMBL7649721 0.77 ITGB3 (0.45) ITGB3ITGA2BITGAVITGB1ITGB5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6451800-B1 Phenylpiperazine derivatives as integrin αvβ3 antagonists MEIJI SEIKA KAISHA, LTD. (JP) 2002-09-17 US claimed
EP-1057818-A1 PHENYLPIPERAZINE DERIVATIVES AS INTEGRIN ALPHAvBETA3 ANTAGONISTS MEIJI SEIKA KAISHA LTD. (JP) 2000-12-06 EP claimed
US-6451800-B1 Phenylpiperazine derivatives as integrin αvβ3 antagonists MEIJI SEIKA KAISHA, LTD. (JP) 2002-09-17 US disclosed
EP-1057818-A1 PHENYLPIPERAZINE DERIVATIVES AS INTEGRIN ALPHAvBETA3 ANTAGONISTS MEIJI SEIKA KAISHA LTD. (JP) 2000-12-06 EP disclosed