SCHEMBL7655014

SCHEMBL7655014

CC(C)Oc1ccc(C(=O)Nc2ccc3c(c2)C(C)N(C)CC3(C)C)cc1C#N

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
NPC1 O15118 1/20 0.39
TP53 P04637 1/20 0.39
RAB9A P51151 1/20 0.39
NPY2R P49146 1/20 0.39
PTGDR2 Q9Y5Y4 1/20 0.39
S1PR1 P21453 2/20 0.38
S1PR3 Q99500 1/20 0.38
XDH P47989 1/20 0.38
EZH2 Q15910 1/20 0.37
RORC P51449 1/20 0.37
MAPT P10636 2/20 0.37
MAPK1 P28482 1/20 0.37
ROCK2 O75116 1/20 0.37
MEN1 O00255 1/20 0.36
HPGD P15428 1/20 0.36
KMT2A Q03164 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
HSD17B10 Q99714 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7656812 0.87 CYP26A1 (0.38) ALDH1A1SMN1; SMN2NPC1RAB9ARORC
SCHEMBL7653578 0.86 RORC (0.47) ALDH1A1SMN1; SMN2NPC1TP53RAB9A
SCHEMBL7655775 0.84 ROCK2 (0.46) ALDH1A1SMN1; SMN2NPC1TP53RAB9A
SCHEMBL7655182 0.79 ROCK2 (0.42) S1PR1S1PR3ROCK2
Hydrochloric Acid SCHEMBL6293630 0.76 ROCK2 (0.57) S1PR1ROCK2
SCHEMBL7658675 0.76 ROCK2 (0.42) TP53NPY2RS1PR1ROCK2
SCHEMBL7654514 0.76 MAPT (0.56) ALDH1A1SMN1; SMN2NPC1TP53MAPT
SCHEMBL7660384 0.76 ROCK2 (0.51) ALDH1A1SMN1; SMN2NPC1RAB9AMAPT
SCHEMBL7649851 0.76 MAPT (0.49) SMN1; SMN2TP53MAPTROCK2MEN1
SCHEMBL7009661 0.74 RORC (0.49) NPY2RRORCROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6492378-B1 Substituted isoquinoline derivatives and their use as anticonvulsivants SMITHKLINE BEECHAM P.L.C. (GB) 2002-12-10 US disclosed