SCHEMBL7655100

SCHEMBL7655100

COc1ccc(Cn2c(=O)[nH]c3cc([N+](=O)[O-])ccc3c2=O)cc1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.65
GAA P10253 5/20 0.56
TP53 P04637 2/20 0.56
ALDH1A1 P00352 5/20 0.55
HTT P42858 3/20 0.54
HSD17B10 Q99714 3/20 0.54
SMN1; SMN2 Q16637 2/20 0.54
USP2 O75604 1/20 0.54
LMNA P02545 1/20 0.54
PKM P14618 1/20 0.54
TSHR P16473 1/20 0.54
CASP1 P29466 1/20 0.54
CASP7 P55210 1/20 0.54
NPSR1 Q6W5P4 1/20 0.54
MAPT P10636 4/20 0.52
MEN1 O00255 3/20 0.52
KMT2A Q03164 3/20 0.52
L3MBTL1 Q9Y468 1/20 0.52
HTR3A P46098 1/20 0.52
RXFP1 Q9HBX9 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7650431 0.91 KDM4E (0.65) KDM4EGAATP53MEN1KMT2A
SCHEMBL7655012 0.82 KDM4E (0.72) KDM4EGAATP53ALDH1A1HTT
SCHEMBL7985041 0.82 KMT2A (0.53) KDM4EALDH1A1SMN1; SMN2MAPTMEN1
SCHEMBL17242598 0.81 KDM4E (0.70) KDM4EGAATP53ALDH1A1HTT
SCHEMBL4254375 0.79 ALDH1A1 (0.72) KDM4EGAATP53ALDH1A1HTT
SCHEMBL7593290 0.78 MEN1 (0.77) KDM4EGAATP53ALDH1A1HTT
SCHEMBL28694312 0.78 KDM4E (0.56) KDM4ETP53ALDH1A1HSD17B10SMN1; SMN2
SCHEMBL29428154 0.78 KDM4E (0.56) KDM4ETP53ALDH1A1HSD17B10SMN1; SMN2
SCHEMBL17242517 0.78 KDM4E (0.76) KDM4EGAATP53ALDH1A1HTT
SCHEMBL4256455 0.78 GAA (0.72) KDM4EGAATP53ALDH1A1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6407116-B1 2,4-DIOXO-1,2,3,4-TETRAHYDROQUINAZOLINE DERIVATIVES; ANTIALLERGENS, ANTIASTHMATICS, ANTIHISTAMINES, AND ANTIINFLAMMATORY AGENTS TAKEDA CHEMICAL INDUSTRIES, INC. (JP) 2002-06-18 US disclosed
EP-1026160-A1 NITROGENOUS FUSED-RING COMPOUNDS, PROCESS FOR THE PREPARATION OF THE SAME, AND DRUGS Takeda Chemical Industries, Ltd. (JP) 2000-08-09 EP disclosed