SCHEMBL7656241

SCHEMBL7656241

CSCC[C@](C)(NC(=O)c1ccc(NC(Cn2ccnc2)c2ccc(F)cc2)cc1-c1ccc(F)cc1)C(=O)O

nearest known ligand 0.40

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CYP51A1 Q16850 6/20 0.40
PTGS2 P35354 1/20 0.39
CYP3A4 P08684 3/20 0.38
CYP2C19 P33261 3/20 0.38
CYP2D6 P10635 2/20 0.38
CYP2C9 P11712 2/20 0.38
FNTA P49354 4/20 0.37
FNTB P49356 4/20 0.37
PGGT1B P53609 1/20 0.35
CYP1A2 P05177 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7667482 0.97 PTGS2 (0.43) CYP51A1PTGS2CYP3A4CYP2C19CYP2D6
SCHEMBL7660603 0.91 PTGS2 (0.40) CYP51A1PTGS2CYP3A4CYP2C19CYP2D6
SCHEMBL7662081 0.89 CYP51A1 (0.40) CYP51A1PTGS2CYP3A4CYP2C19CYP2D6
SCHEMBL7657941 0.88 FNTA (0.37) CYP51A1PTGS2CYP3A4CYP2C19CYP2D6
SCHEMBL7561783 0.85 PTGS2 (0.43) CYP51A1PTGS2CYP3A4CYP2C19CYP2D6
SCHEMBL7585240 0.85 PTGS2 (0.43) CYP51A1PTGS2CYP3A4CYP2C19CYP2D6
SCHEMBL7654320 0.84 FNTA (0.53) FNTAFNTBPGGT1B
SCHEMBL7561794 0.83 FNTA (0.40) CYP51A1PTGS2CYP3A4CYP2C19CYP2D6
SCHEMBL8211342 0.82 FNTA (0.42) CYP51A1PTGS2CYP3A4CYP2C19CYP2D6
SCHEMBL7660388 0.81 FNTA (0.56) FNTAFNTBPGGT1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6410539-B1 ANTICARCINOGENIC AGENTS ASTRAZENCA UK LIMITED (GB) 2002-06-25 US claimed