SCHEMBL7656636

SCHEMBL7656636

O=C(NCC(O)CO)c1ccc(C(=O)NCC(O)CO)nc1

nearest known ligand 0.50

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.47
KDM4E B2RXH2 2/20 0.47
HPGD P15428 1/20 0.47
GABRA5 P31644 1/20 0.47
PRMT5 O14744 3/20 0.46
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
P4HTM Q9NXG6 2/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
MAOB P27338 1/20 0.40
MAP2K1 Q02750 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7663932 0.87 ALDH1A1 (0.44) ALDH1A1KDM4EPRMT5NPC1RAB9A
SCHEMBL7661497 0.86 ALDH1A1 (0.46) ALDH1A1KDM4ENPC1RAB9AP4HTM
SCHEMBL6388225 0.84 HDAC1 (0.49) ALDH1A1KDM4ENPC1RAB9AP4HTM
SCHEMBL7105165 0.84 MAP2K1 (0.41) ALDH1A1KDM4EHPGDMAP2K1
SCHEMBL8824679 0.84 THRB (0.54) ALDH1A1KDM4ENPC1RAB9AP4HTM
SCHEMBL24336711 0.80 GABRA5 (0.44) ALDH1A1KDM4EHPGDGABRA5PRMT5
SCHEMBL21365172 0.80 GABRA5 (0.44) ALDH1A1KDM4EHPGDGABRA5PRMT5
SCHEMBL19878599 0.80 GABRA5 (0.44) ALDH1A1KDM4EHPGDGABRA5PRMT5
SCHEMBL19878598 0.80 GABRA5 (0.44) ALDH1A1KDM4EHPGDGABRA5PRMT5
SCHEMBL8061648 0.80 ALDH1A1 (0.42) ALDH1A1KDM4EGABRA5PRMT5NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6399613-B1 N,N'-BIS(2-HYDROXYETHYL)PYRAZINE-2,5- OR -2,6-DICARBOXAMIDE; DIABETES AVENTIS PHARMA S.A. (FR) 2002-06-04 US claimed
US-6399613-B1 N,N'-BIS(2-HYDROXYETHYL)PYRAZINE-2,5- OR -2,6-DICARBOXAMIDE; DIABETES AVENTIS PHARMA S.A. (FR) 2002-06-04 US disclosed