SCHEMBL7657510

SCHEMBL7657510

O=C(NC(O)CCO)c1ccc(C(=O)NC(O)CCO)nc1

nearest known ligand 0.45

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.45
KDM4E B2RXH2 1/20 0.45
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
MME P08473 2/20 0.41
P4HTM Q9NXG6 6/20 0.40
LMNA P02545 2/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
POLB P06746 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
AHR P35869 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7658593 0.84 CNR2 (0.38) ALDH1A1NPC1RAB9AMMELMNA
SCHEMBL7655301 0.82 ALDH1A1 (0.43) ALDH1A1KDM4ENPC1RAB9AMME
SCHEMBL7657495 0.80 ALDH1A1 (0.49) ALDH1A1KDM4ENPC1RAB9AMME
SCHEMBL7655289 0.78 ALDH1A1 (0.44) ALDH1A1KDM4ENPC1RAB9AMME
SCHEMBL13164714 0.76 GRM5 (0.56) ALDH1A1KDM4ENPC1RAB9AP4HTM
SCHEMBL28453112 0.74 FOLH1 (0.44)
SCHEMBL7659871 0.74 LMNA (0.45) ALDH1A1KDM4ELMNAMEN1KMT2A
SCHEMBL7653658 0.74 KDM4E (0.44) ALDH1A1KDM4EPOLB
SCHEMBL7650766 0.74 CTSA (0.35) LMNA
SCHEMBL13210632 0.74 ALDH1A1 (0.55) ALDH1A1KDM4ENPC1RAB9AP4HTM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6399613-B1 N,N'-BIS(2-HYDROXYETHYL)PYRAZINE-2,5- OR -2,6-DICARBOXAMIDE; DIABETES AVENTIS PHARMA S.A. (FR) 2002-06-04 US claimed
US-6399613-B1 N,N'-BIS(2-HYDROXYETHYL)PYRAZINE-2,5- OR -2,6-DICARBOXAMIDE; DIABETES AVENTIS PHARMA S.A. (FR) 2002-06-04 US disclosed