Prometryn

Prometryn

SCHEMBL7657627

CSc1nc(NC(C)C)nc(NC(C)C)n1.CSc1nc(NC(C)C)nc(NC(C)C)n1

nearest known ligand 0.56

Full drug profile on Sugi Atlas →

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 3/20 0.56
GAA P10253 5/20 0.54
TDP1 Q9NUW8 2/20 0.54
HTT P42858 3/20 0.48
LMNA P02545 2/20 0.48
F2 P00734 1/20 0.48
SMN1; SMN2 Q16637 2/20 0.48
TSHR P16473 1/20 0.48
HSD17B10 Q99714 1/20 0.48
KMT2A Q03164 4/20 0.47
ALDH1A1 P00352 4/20 0.47
KDM4E B2RXH2 1/20 0.47
MEN1 O00255 2/20 0.45
CYP1A2 P05177 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
KCNH3 Q9ULD8 2/20 0.44
MAPT P10636 1/20 0.41
CYP2C9 P11712 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Prometryn SCHEMBL7622 1.00 MAPK1 (0.56) MAPK1GAATDP1HTTLMNA
Prometryn SCHEMBL20723889 0.98 GAA (0.58) MAPK1GAATDP1HTTLMNA
SCHEMBL29435432 0.92 MAPK1 (0.50) MAPK1GAATDP1HTTLMNA
SCHEMBL66639 0.92 MAPK1 (0.50) MAPK1GAATDP1HTTLMNA
SCHEMBL8827500 0.92 MAPK1 (0.50) MAPK1GAATDP1HTTLMNA
Prometryn SCHEMBL5542826 0.88 TSHR (0.48) MAPK1GAATDP1HTTLMNA
SCHEMBL24059309 0.87 MAPK1 (0.50) MAPK1GAATDP1HTTLMNA
Prometryn SCHEMBL7945620 0.87 POLB (0.54) MAPK1GAAHTTLMNATSHR
Ametryne SCHEMBL8541067 0.87 POLB (0.54) MAPK1GAAHTTLMNATSHR
Ametryne SCHEMBL65196 0.87 POLB (0.54) MAPK1GAAHTTLMNATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 69 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0009620-B1 HERBICIDES AND THEIR APPLICATION TO THE CONTROL OF WEEDS HOECHST AKTIENGESELLSCHAFT (DE) 1981-08-05 EP claimed
EP-0009620-A1 Herbicides and their application to the control of weeds HOECHST AKTIENGESELLSCHAFT (DE) 1980-04-16 EP claimed
EP-1223988-A1 ANTISENSE MODULATION OF TUMOR NECROSIS FACTOR ALPHA CONVERTING ENZYME (TACE) EXPRESSION ISIS PHARMACEUTICALS, INC. (US) 2002-07-24 EP disclosed
WO-2001030360-A1 MODULATION OF L-SELECTIN SHEDDING VIA INHIBITION OF TUMOR NECROSIS FACTOR ALPHA CONVERTING ENZYME (TACE) ISIS PHARMACEUTICALS, INC. (US) 2001-05-03 WO disclosed
WO-2001030395-A1 ANTISENSE MODULATION OF TUMOR NECROSIS FACTOR ALPHA CONVERTING ENZYME (TACE) EXPRESSION ISIS PHARMACEUTICALS, INC. (US) 2001-05-03 WO disclosed
EP-0902681-A1 INHIBITION OF SELECTIN BINDING THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1999-03-24 EP disclosed
EP-0574418-B1 ARYL SULPHONYL UREA COMPOUNDS, A METHOD OF PREPARING THEM, AND THEIR USE AS HERBICIDES AND GROWTH REGULATORS HOECHST SCHERING AGREVO GMBH (DE) 1998-11-11 EP disclosed
US-5688745-A Arylsulfonylureas and their use as herbicides and growth regulators HOECHST AKTIENGESELLSCHAFT (DE) 1997-11-18 US disclosed
WO-1997031625-A1 INHIBITION OF SELECTIN BINDING THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1997-09-04 WO disclosed
US-5463081-A Chemical intermediates HOECHST AKTIENGESELLSCHAFT (DE) 1995-10-31 US disclosed
WO-1992020684-A1 HERBICIDAL OXATRICYCLIC ETHERS E.I. DU PONT DE NEMOURS AND COMPANY (US) 1992-11-26 WO disclosed
US-4278613-A ANTIDOTES CIBA-GEIGY CORPORATION (US) 1981-07-14 US disclosed
US-4269775-A DERIVATIVES OF PHENYL OR NAPHTHYL ACETONITRILE OXIME-ALKYLENE-DIETHERS; ANTIDOTES FOR HERBICIDES CIBA-GEIGY CORPORATION (US) 1981-05-26 US disclosed
EP-0019796-A1 Propionic acid esters, preparation of these compounds, herbicides containing these compounds as active substances, and the use of such compounds and agents for combating weeds F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1980-12-10 EP disclosed
EP-0012158-A2 Oxime derivatives and their use in the protection of cultivated plants CIBA-GEIGY AG (CH) 1980-06-25 EP disclosed
EP-0010588-A2 Sulfur-containing oxime compounds and their use to protect cultivated plants CIBA-GEIGY AG (CH) 1980-05-14 EP disclosed
EP-0011047-A2 Oxime derivatives to protect cultivated plants CIBA-GEIGY AG (CH) 1980-05-14 EP disclosed
EP-0010143-A2 Oxime derivatives to protect cultivated plants CIBA-GEIGY AG (CH) 1980-04-30 EP disclosed
EP-0010058-A1 Process and compositions for the protection of plant cultures against the phytotoxic action of strong herbicides; oxime ether derivatives CIBA-GEIGY AG (CH) 1980-04-16 EP disclosed
EP-0009620-A1 Herbicides and their application to the control of weeds HOECHST AKTIENGESELLSCHAFT (DE) 1980-04-16 EP disclosed