SCHEMBL7657754

SCHEMBL7657754

NOC(=O)CCNC(=O)c1ccc(N2CCN(c3ncccn3)CC2)cc1

nearest known ligand 0.58

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.58
HTT P42858 1/20 0.58
RAB9A P51151 2/20 0.53
NPC1 O15118 1/20 0.53
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47
CA7 P43166 1/20 0.47
CA9 Q16790 1/20 0.47
HDAC6 Q9UBN7 3/20 0.47
ALDH1A1 P00352 1/20 0.44
GFER P55789 1/20 0.44
DRD2 P14416 1/20 0.44
MAPT P10636 1/20 0.43
KMT2A Q03164 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7539336 0.90 KDM4E (0.60) KDM4EHTTRAB9ANPC1CA1
SCHEMBL7655831 0.87 KDM4E (0.56) KDM4EHTTRAB9ANPC1CA1
SCHEMBL7655169 0.86 KDM4E (0.67) KDM4EHTTRAB9ANPC1CA1
SCHEMBL7655246 0.83 KDM4E (0.50) KDM4EHTTALDH1A1DRD2KMT2A
SCHEMBL382963 0.83 SMYD3 (0.43) KDM4EHTTALDH1A1GFERDRD2
SCHEMBL7655291 0.81 KDM4E (0.53) KDM4EHTTRAB9ANPC1HDAC6
SCHEMBL7658795 0.81 KDM4E (0.55) KDM4EHTTRAB9ANPC1CA1
SCHEMBL6375221 0.80 RAB9A (0.67) KDM4EHTTRAB9ANPC1CA1
SCHEMBL7657964 0.79 KDM4E (0.52) KDM4EHTTRAB9ANPC1CA1
SCHEMBL7049509 0.78 ITGB3 (0.42) KDM4EHTTRAB9ANPC1HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6451800-B1 Phenylpiperazine derivatives as integrin αvβ3 antagonists MEIJI SEIKA KAISHA, LTD. (JP) 2002-09-17 US claimed
EP-1057818-A1 PHENYLPIPERAZINE DERIVATIVES AS INTEGRIN ALPHAvBETA3 ANTAGONISTS MEIJI SEIKA KAISHA LTD. (JP) 2000-12-06 EP claimed
US-6451800-B1 Phenylpiperazine derivatives as integrin αvβ3 antagonists MEIJI SEIKA KAISHA, LTD. (JP) 2002-09-17 US disclosed
EP-1057818-A1 PHENYLPIPERAZINE DERIVATIVES AS INTEGRIN ALPHAvBETA3 ANTAGONISTS MEIJI SEIKA KAISHA LTD. (JP) 2000-12-06 EP disclosed