SCHEMBL7657964

SCHEMBL7657964

O=C(CCNC(=O)c1ccc(N2CCCN(c3ncccn3)CC2)cc1)ONS(=O)(=O)c1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.52
HTT P42858 1/20 0.52
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
CA7 P43166 1/20 0.43
CA9 Q16790 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
ITGB3 P05106 1/20 0.42
ITGA2B P08514 1/20 0.42
ALDH1A1 P00352 1/20 0.42
LMNA P02545 1/20 0.42
MAPK1 P28482 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
HTR1A P08908 1/20 0.41
ADRA2A P08913 1/20 0.41
ADRA2B P18089 1/20 0.41
ADRA2C P18825 1/20 0.41
ADRA1D P25100 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7658795 0.97 KDM4E (0.55) KDM4EHTTCA1CA2CA7
SCHEMBL7463691 0.88 KDM4E (0.52) KDM4EHTTHDAC6RAB9AALDH1A1
SCHEMBL7653652 0.85 KDM4E (0.44) KDM4EHTTITGB3ITGA2BHTR1A
SCHEMBL7652415 0.85 KDM4E (0.44) KDM4EHTTITGB3ITGA2BHTR1A
SCHEMBL7652041 0.85 KDM4E (0.44) KDM4EHTTITGB3ITGA2BHTR1A
SCHEMBL7654976 0.84 KDM4E (0.44) KDM4EHTTITGB3ITGA2BLMNA
SCHEMBL7658560 0.84 KDM4E (0.48) KDM4EHTTITGB3ITGA2BALDH1A1
SCHEMBL7654380 0.84 DRD2 (0.44) KDM4EHTTALDH1A1LMNAMAPK1
SCHEMBL7653683 0.84 KDM4E (0.44) KDM4EHTTITGB3ITGA2BALDH1A1
SCHEMBL382763 0.83 ITGB3 (0.48) KDM4EHTTITGB3ITGA2BHTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1057818-A1 PHENYLPIPERAZINE DERIVATIVES AS INTEGRIN ALPHAvBETA3 ANTAGONISTS MEIJI SEIKA KAISHA LTD. (JP) 2000-12-06 EP claimed
US-6451800-B1 Phenylpiperazine derivatives as integrin αvβ3 antagonists MEIJI SEIKA KAISHA, LTD. (JP) 2002-09-17 US disclosed
EP-1057818-A1 PHENYLPIPERAZINE DERIVATIVES AS INTEGRIN ALPHAvBETA3 ANTAGONISTS MEIJI SEIKA KAISHA LTD. (JP) 2000-12-06 EP disclosed