SCHEMBL7657838

SCHEMBL7657838

CC(=O)Nc1ccc(Cl)c2c1C(=O)CCS2

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.38
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
CA9 Q16790 1/20 0.37
KDM4E B2RXH2 3/20 0.36
HSD17B10 Q99714 2/20 0.36
MAOA P21397 1/20 0.35
GAA P10253 1/20 0.35
HPGD P15428 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
ROCK2 O75116 1/20 0.34
PDE3B Q13370 1/20 0.34
PDE3A Q14432 1/20 0.34
MAPT P10636 2/20 0.33
CASP3 P42574 1/20 0.33
NPC1 O15118 1/20 0.33
POLB P06746 1/20 0.33
RAB9A P51151 1/20 0.33
ATAD2 Q6PL18 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9404925 0.84 POLB (0.41) ALDH1A1CA1CA2CA9KDM4E
SCHEMBL7664272 0.84 ALDH1A1 (0.39) ALDH1A1KDM4EHSD17B10MAOAGAA
SCHEMBL7653076 0.83 HDAC1 (0.38) ALDH1A1CA1CA2CA9KDM4E
SCHEMBL9404817 0.82 MAPT (0.43) ALDH1A1KDM4EGAAHPGDMEN1
SCHEMBL9404941 0.81 ALDH1A1 (0.43) ALDH1A1KDM4EGAAHPGDMEN1
SCHEMBL9404931 0.80 MAOA (0.33) ALDH1A1CA1CA2CA9KDM4E
SCHEMBL9404879 0.80 ALDH1A1 (0.36) ALDH1A1KDM4EHSD17B10MAOAGAA
SCHEMBL7661312 0.79 HDAC1 (0.38) ALDH1A1CA1CA2CA9KDM4E
SCHEMBL9404756 0.78 KCNH2 (0.39) ALDH1A1KDM4EMAOAGAAMEN1
SCHEMBL9404891 0.78 TSHR (0.36) MAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6407115-B1 ANTICARCINOGENIC AND ANTITUMOR AGENTS; SIDE EFFECT REDUCTION, WATER SOLUBILITY DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2002-06-18 US disclosed
US-5834476-A DERIVATIVE OF CAMPTOTHECIN, ANTITUMOR AGENT, ANTICARCINOGENIC AGENT DAIICHI PHARMACEUTICAL CO., LTD. (JP) 1998-11-10 US disclosed
US-5770605-A Method for treating leukemia with a hexa-cyclic compound DAIICHI PHARMACEUTICAL CO., LTD. (JP) 1998-06-23 US disclosed
US-5658920-A ANTITUMOR AGENTS DAIICHI PHARMACEUTICAL CO., LTD. (JP) 1997-08-19 US disclosed
US-5637770-A Hexa-cyclic compound DAIICHI PHARMACEUTICAL CO., LTD. (JP) 1997-06-10 US disclosed
EP-0495432-B1 Hexa-cyclic compound DAIICHI SEIYAKU CO (JP) 1996-05-29 EP disclosed
EP-0495432-A1 Hexa-cyclic compound DAIICHI PHARMACEUTICAL CO., LTD. (JP) 1992-07-22 EP disclosed